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5-methyl-1-(3-methylphenyl)-4-[3-(piperidin-1-yl)propanoyl]piperazin-2-one
(2S,4S)-N-ethyl-4-(4-fluorobenzamido)-1-(thiophen-3-ylmethyl)pyrrolidine-2-carboxamide
2-{1-[(6-methylpyridin-2-yl)methyl]-4-[1-(2-phenylethyl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
(1-{[1-(quinoxaline-6-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
9-[2-(benzenesulfonyl)ethyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-{1-[2-(4-methoxyphenoxy)ethyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
(3S,5R)-5-[(pyridin-2-ylmethyl)carbamoyl]-1-(1H-pyrrole-2-carbonyl)piperidine-3-carboxylic acid
5-[4-(piperidin-1-ylmethyl)benzoyl]-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
1-{2-[1-(2,5-dimethylphenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]ethyl}-5-methyl-1H-1,2,3,4-tetrazole
N-(2,3-dimethylquinoxalin-6-yl)-4-(1H-pyrrole-2-carbonyl)piperazine-1-carboxamide
1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
(3S,4S)-1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-4-(piperidin-1-yl)pyrrolidin-3-ol
methyl 9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-3-[2-(2-methylphenyl)acetyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-chloro-4-fluoro-N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)benzamide
7-[2-(2-chloro-4-fluorophenoxy)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-{[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]amino}pyridine-3-carbonitrile
4-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-1-(4-fluorophenyl)butan-1-one
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2,4-dimethyl-1,3-oxazole-5-carboxamide
N-(1-benzyl-1H-pyrazol-3-yl)-2-[3-(4-methylthiophen-2-yl)-1H-pyrazol-1-yl]acetamide
1-(2-aminoethyl)-N-{[1-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-2-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
1-(2-methoxypyridine-3-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
1-(cyclobutylmethyl)-3-({[(3-fluorophenyl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
1-[2-(dimethylamino)-4-(4-hydroxypiperidin-1-yl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]-3-hydroxypropan-1-one
N'1-[2-(3-phenylpropoxy)phenyl]cyclopropane-1,1-dicarboxamide
6-[2-(diethylamino)ethyl]-5,6-dihydro-1,6-naphthyridin-5-one
ethyl 1-{2-[4-(3-phenoxypropanamido)-1H-pyrazol-1-yl]acetyl}piperidine-3-carboxylate
N-cyclopropyl-5-(3-acetamidophenyl)thiophene-2-carboxamide
5-(propan-2-yl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}-1,2-oxazole-3-carboxamide
N-{2-[4-(furan-2-ylmethyl)morpholin-2-yl]ethyl}-3-methylthiophene-2-carboxamide
4-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}-2-(trifluoromethyl)morpholine
2-[1-cyclopentyl-4-(quinolin-2-ylmethyl)piperazin-2-yl]ethan-1-ol
2-{1-cyclohexyl-4-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-(4-chloro-2-{7-oxo-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-5-yl}phenoxy)acetic acid
[(3S,5R)-1-(2,6-dimethoxypyridine-3-carbonyl)-5-[(dimethylamino)methyl]piperidin-3-yl]methanol
[2-methoxy-5-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenyl]methanol
N-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}-2-methyl-1H-1,3-benzodiazole-4-carboxamide
4-methyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-3-phenyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
1-[(2-fluorophenyl)methyl]-4-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}-1,4-diazepane
2-ethyl-4-methyl-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1,3-oxazole-5-carboxamide
5-(4-methanesulfonylpiperazine-1-carbonyl)-4-methyl-2-(pyridin-3-yl)pyrimidine
N4,N4,5-trimethyl-N2-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]pyrimidine-2,4-diamine
5-methanesulfonyl-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-4-(piperidin-3-yl)pyrimidin-2-amine
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-2-(pyridin-3-yl)pyridine
4-{1-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-yl}benzoic acid
(3R,4S)-N,N-dimethyl-4-(5-methylfuran-2-yl)-1-(oxane-4-carbonyl)pyrrolidin-3-amine
propan-2-yl 2-chloro-5-(3,5-dimethyl-4,5-dihydro-1,2-oxazole-5-amido)benzoate
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-(piperidine-1-sulfonyl)pyrrolidin-3-yl]methanol
(2S,4R)-4-(4-{[(tert-butylcarbamoyl)(methyl)amino]methyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
5-{[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)methyl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
5-propyl-2-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl}pyrimidine