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2-(ethylamino)-N-[(3R,4R)-4-(4-methylpiperazin-1-yl)oxolan-3-yl]pyrimidine-5-carboxamide
N-(2-methoxy-2-methylpropyl)-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
3-(4-fluorophenoxymethyl)-1-(propan-2-yl)-5-[2-(trimethyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,4-triazole
1-(1-benzofuran-5-carbonyl)-4-(benzyloxy)piperidine
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]acetic acid
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-(2-methylquinolin-4-yl)pyrrolidin-3-yl]methanol
6-(2-butoxy-4-fluorophenyl)-2-methyl-2,3-dihydropyridazin-3-one
(1R,5R)-6-(2,3-dimethylquinoxaline-6-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1,5-dimethyl-2-phenyl-4-{1-[1-(pyrimidin-4-yl)ethyl]-1H-imidazol-2-yl}-2,3-dihydro-1H-pyrazol-3-one
4-methoxy-N-({1-[2-(piperidin-1-yl)acetyl]piperidin-3-yl}methyl)benzene-1-sulfonamide
1-[2-methyl-2-(morpholin-4-yl)propyl]-4-(3-methylpyridin-4-yl)-1,4-diazepane
N-methyl-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-(1-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-pyrazol-4-yl)ethan-1-ol
6-{2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-2-carbonitrile
(1R,2S,9R)-11-{5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carbonyl}-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
5-fluoro-2-{4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}-1H-indole
7-[(4-ethyl-1,3-thiazol-2-yl)methyl]-2-oxa-7-azaspiro[4.5]decan-8-one
2-[(4-cyclopentylpyrimidin-2-yl)amino]-N-methylethane-1-sulfonamide
2-(4-butyl-3-oxopiperazin-1-yl)-N-cyclopentylpropanamide
1-[3-(pyrrolidin-1-yl)propyl]-4-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1,4-diazepane
N-(1H-imidazol-2-ylmethyl)-1-methyl-N-(pyridin-3-ylmethyl)piperidin-4-amine
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-4-(2-oxopyrrolidin-1-yl)benzamide
1-[4-(furan-2-yl)phenyl]-3-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]urea
(1R,9S)-5-amino-3-(1-benzofuran-2-yl)-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
methyl({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})[2-(oxan-2-yl)ethyl]amine
(1S,6R)-3-{2-[4-(2-fluorophenyl)piperazin-1-yl]-2-oxoethyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
1-[(4-methoxyphenyl)methyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
methyl 6-[(3S,4R)-3-methanesulfonamido-4-(propan-2-yl)pyrrolidin-1-yl]pyrimidine-4-carboxylate
2-(pyridin-3-ylmethyl)-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
2-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]benzene-1,3-diol
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
(4aS,7aR)-1-{[2-(2-hydroxyethoxy)phenyl]methyl}-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-2-methyl-1-benzofuran-7-carboxamide
(3S,9aR)-8-(3-fluoro-4-methylbenzoyl)-3-[(1R)-1-hydroxyethyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{4-[2-(2,3-dimethylphenoxy)ethyl]piperazin-1-yl}pyridine-3-carbonitrile
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-3-chlorobenzamide
N-{[3-(dimethylamino)thiolan-3-yl]methyl}-2-(methylamino)pyridine-4-carboxamide
2-(4-methoxy-3,5-dimethylphenyl)-2-({[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)amino)acetic acid
N-benzyl-1-{2-[(2,4-dimethoxyphenyl)formamido]ethyl}-N-methyl-1H-1,2,3-triazole-4-carboxamide
5,6-dimethyl-2-[5-(oxolane-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-1H-1,3-benzodiazole
1-[2-methoxy-5-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)phenoxy]-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
N-(4-methoxy-2-methylphenyl)-3-[1-(1,2,4-oxadiazol-3-ylmethyl)piperidin-3-yl]propanamide
2-{[2-(2-hydroxyethyl)morpholin-4-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
3-(1H-imidazol-1-ylmethyl)-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidine
3-{1-[1-(3-aminopropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(3-fluorophenyl)urea
(1S,5R)-6-[(2,3-difluoro-6-methoxyphenyl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-{[8-methoxy-2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}phenol
6-{[1-(4-acetylpiperazin-1-yl)hex-5-en-2-yl]oxy}pyridine-2-carbonitrile
(1R,5R)-N,N-dimethyl-6-[2-(pyridin-4-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-(2-hydroxyethyl)-2-[(2-methylprop-2-en-1-yl)oxy]-N-(1,3-thiazol-2-ylmethyl)benzamide