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1-benzyl-4-(4-methylpent-3-en-1-yl)-1,4-diazepan-6-ol
N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3,5-dimethylbenzamide
2-[1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)pyrrolidin-2-yl]pyridine
2-methoxy-N-[2-methoxy-5-({[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]carbamoyl}amino)phenyl]acetamide
5-{[(2,4-difluorophenyl)methyl]amino}-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(4-methyl-1H-pyrrole-2-carbonyl)-3-(4-methylphenoxymethyl)piperidine
{[2-(4-methoxyphenyl)-7-methylquinolin-3-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
ethyl 3-[(2E)-3-phenylprop-2-en-1-yl]-1-[2-(1H-pyrazol-1-yl)acetyl]piperidine-3-carboxylate
N2-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-N4-methylpyrimidine-2,4-diamine
3-(2-fluorophenyl)-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-3-phenylpropanamide
4-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-N-methyl-4-oxobutanamide
2-[2-(1-benzofuran-2-yl)-1H-imidazol-1-yl]-N-(2-methylphenyl)acetamide
(3aS,7aR)-5-methyl-2-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
3-(5-{[4-(difluoromethoxy)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
1-(cyclopropylmethyl)-5-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
methyl[(4-methyl-1H-imidazol-5-yl)methyl]{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}amine
2-methyl-5-phenyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
N-(2-methylphenyl)-3-{[6-(piperidin-3-yl)pyrimidin-4-yl]amino}propanamide
2-methyl-7-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-[1,3]oxazolo[5,4-d]pyrimidine
methyl[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl](thiophen-3-ylmethyl)amine
4-cyano-1-methyl-N-[1-(pyrrolidin-1-ylmethyl)cyclohexyl]-1H-pyrrole-2-carboxamide
[(3R,4R)-1-[2-amino-6-(methylamino)pyrimidin-4-yl]-4-(azepan-1-ylmethyl)pyrrolidin-3-yl]methanol
4-(1H-imidazol-1-ylmethyl)-1-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-ol
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
5-{4-[(2-fluorophenyl)methyl]piperidine-1-carbonyl}-2,2-dimethylthiomorpholin-3-one
1-(1-benzylpiperidin-4-yl)-3-(4-chlorobenzoyl)piperidine
7-methoxy-N,N-dimethyl-2-[1-(3-methylpyridin-4-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
2-(1-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}piperidin-2-yl)pyridine
2-(2,3-difluorophenoxymethyl)-N-[2-(pyrazin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
3-[2-(pyrrolidine-1-sulfonyl)ethyl]-1-[3-(1,3-thiazol-4-yl)phenyl]urea
1-(1-methyl-5-{[(1R,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1H-pyrrol-3-yl)ethan-1-one
4,6-dimethyl-2-[4-(pyrrolidine-1-carbonyl)phenyl]pyrimidine
2-methyl-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyridine-3-carboxamide
methyl 4-[(2-{[4-(pyridin-3-yloxy)phenyl]carbamoyl}piperidin-1-yl)methyl]benzoate
3-[(4-ethylphenyl)methyl]-N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
3-[(3R,4S)-4-(morpholin-4-yl)-1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-yl]propan-1-ol
1-[(2-fluorophenyl)methyl]-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
5-({[(3-{2-[4-(5-fluoro-2-methylbenzenesulfonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
4-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-N-propylbenzene-1-sulfonamide
5-{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-(2-fluoro-4-methoxyphenyl)-2-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
6-(2H-1,3-benzodioxole-5-carbonyl)-3-(4-fluoro-3-methylphenyl)-1-(pyridin-3-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-(cyclopent-1-ene-1-carbonyl)-N-phenylpiperidin-3-amine
3-(2-chlorophenyl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
4-(hydroxymethyl)-1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperidin-4-ol
N-[2-(2,5-dimethylphenoxy)ethyl]-N-methyl-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide