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9-[1-(4-chlorophenyl)cyclobutanecarbonyl]-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
N-[(1R,3S)-3-(thiomorpholine-4-carbonyl)cyclopentyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
3-amino-1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propan-1-one
(3R,4S)-3,4-dimethyl-1-(2-methylpyrimidine-5-carbonyl)piperidin-4-ol
5-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1-[(3-methylphenyl)methyl]-3-(oxolan-3-yl)-1H-1,2,4-triazole
methyl 3-[(2E)-3-(3-fluorophenyl)prop-2-enamido]-6-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
N-[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
8-acetyl-2-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-methyl-4-{4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}benzene-1-sulfonamide
1-{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-5-one
dimethyl(2-{2-[1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
5-acetyl-N-[1-(3-methoxyphenyl)ethyl]-N-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-(cyclopropanesulfonyl)-4-phenoxypiperidine-4-carboxylic acid
1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-4-(thiophen-2-ylmethyl)-1,4-diazepane
2-{2-chloro-4-[(4-ethyl-2-methyl-3-oxopiperazin-1-yl)methyl]-6-methoxyphenoxy}acetic acid
1-{4-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]phenyl}imidazolidine-2,4-dione
methyl 6-[(4-methylpiperidin-1-yl)methyl]-3-(thiophene-3-amido)thieno[2,3-b]pyridine-2-carboxylate
1-[(2-methoxyphenyl)methyl]-N3-methyl-N5-(3-methylbutyl)-4-oxo-N3-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
(2S,4R)-4-amino-N-methyl-1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)pyrrolidine-2-carboxamide
methyl 4-{3-oxo-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-8-yl}butanoate
2-(pyridin-2-ylmethyl)-8-(1,3-thiazol-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
{4-[(3-methoxyphenyl)methyl]-1-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]piperidin-4-yl}methanol
(3aR,6aS)-5-(1-ethyl-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperazine
{[2-(1H-imidazol-2-yl)phenyl]methyl}(methyl)[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]amine
2,3-dioxo-N-[2-(1,3-thiazol-4-yl)ethyl]-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
8-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
(3aR,6aR)-2-(cyclobutylmethyl)-5-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-4-(1H-1,2,3,4-tetrazol-1-yl)phenol
2-{[3-(2-hydroxyethyl)-4-[(4-methylphenyl)methyl]piperazin-1-yl]methyl}phenol
3-[2-(1,4-oxazepan-4-yl)-2-oxoethyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-one
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]acetamide
2-(cyclopropylmethyl)-9-[(4-methoxy-2-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{2-[1-(3,3,3-trifluoropropyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)azepane
2-(4-fluoro-2-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-(3-chloro-4-hydroxyphenyl)-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}acetamide
(1S,5R)-6-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
3-(2-fluorophenyl)-N-(2-methoxyethyl)-N-propyl-1H-pyrazole-4-carboxamide
2-{9-[(2-methyl-1,3-oxazol-4-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
1-[4-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-3,5-dimethyl-1H-pyrrol-2-yl]ethan-1-one
3-[1-(3-chloro-1,2-oxazole-5-carbonyl)piperidin-4-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(4-{[(dimethyl-1,2-oxazol-4-yl)methyl]amino}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
4-[(4-fluorophenyl)methyl]-1-[2-(2-methoxyethoxy)acetyl]-3-(propan-2-yl)-1,4-diazepan-5-one
(1H-imidazol-2-ylmethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)(2-methylpropyl)amine
5-(1-butanoylpiperidin-4-yl)-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
3-{[ethyl({[2-(prop-2-en-1-yloxy)phenyl]methyl})amino]methyl}-7-fluoro-1,2-dihydroquinolin-2-one
2-{5-[2-(dimethylamino)pyrimidin-5-yl]-4-phenyl-1H-imidazol-1-yl}-3-hydroxypropanoic acid
2-(2-{[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
1-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(thiophen-3-yl)ethan-1-one