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8-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-(3-chlorophenyl)-4-(6-ethyl-2-methylpyrimidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-cyclopentyl-3-[2-(methylsulfanyl)benzoyl]piperidine
1-{2-[2-(4-fluorophenyl)piperidin-1-yl]-2-oxoethyl}piperidine-4-carboxamide
[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl](methyl)(oxolan-3-ylmethyl)amine
(4aS,7aR)-1-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[3-(3-methylphenyl)benzoyl]-4-[2-(piperidin-1-yl)ethyl]-1,4-diazepan-5-one
1-(2,6-dimethylpyridin-4-yl)-4-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperazine
N-ethyl-N-[2-phenyl-1-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)ethyl]oxane-4-carboxamide
methyl({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})[3-(1-methyl-1H-imidazol-2-yl)propyl]amine
methyl (1R,3S,3aR,6aS)-1-(2-methoxy-2-oxoethyl)-5-methyl-3-(4-methyl-1H-imidazol-5-yl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
8-(4-methylpiperidine-4-carbonyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
3-methyl-7-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
(1S,3R)-3-(1-butyl-3-cyclopropyl-1H-1,2,4-triazol-5-yl)cyclohexan-1-amine
2-phenoxy-1-{4-[2-(pyridin-2-yl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}propan-1-one
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
(1R,3S)-3-[1-(3-fluorophenyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]cyclopentan-1-amine
N-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
N-butyl-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
(4aS,7aR)-1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-{6-methyl-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carbonyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
2-(5-acetylthiophen-3-yl)-1-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]ethan-1-one
N-(5-methyl-1-propyl-1H-pyrazol-3-yl)-5-({[1-(pyridin-3-yl)propyl]amino}methyl)-1,3-thiazol-2-amine
ethyl 3-[(3-chlorophenyl)methyl]-1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]piperidine-3-carboxylate
1-[1-(2-amino-6-methoxypyrimidin-4-yl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidine
4-[4-(3,4,5-trimethoxyphenyl)phenyl]morpholine
N-benzyl-5-{[(1-hydroxycyclohexyl)methyl]amino}-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-2-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
3-chloro-N-(2-methoxyethyl)-4-({1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}oxy)benzamide
3-(1H-pyrazol-1-ylmethyl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}benzamide
N-[3-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]-4-(4H-1,2,4-triazol-4-yl)piperidine-1-carboxamide
2-methyl-4-{3-[4-(trifluoromethyl)piperidine-1-carbonyl]phenyl}butan-2-ol
1-(6-methoxypyrimidin-4-yl)-N-methyl-N-(2-phenylethyl)piperidin-3-amine
1-(4-{1-azabicyclo[2.2.2]octan-3-yl}piperazin-1-yl)-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
1-(3-ethyl-1,2-oxazole-5-carbonyl)-4-[(3-fluorophenyl)methyl]piperazine
8-{3-methyl-5-[2-(pyridin-3-yl)ethyl]-1H-1,2,4-triazol-1-yl}quinoline
3-amino-N-[1-(3-methylpyridin-2-yl)propyl]-1H-1,2,4-triazole-5-carboxamide
2-{[2-(1H-1,3-benzodiazol-2-yl)ethyl]amino}pyridine-3-carboxamide
1-(2-methoxyphenyl)-5-[(E)-2-(1-methyl-1H-pyrazol-4-yl)ethenyl]-3-(propan-2-yl)-1H-1,2,4-triazole
3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{[4-(hydroxymethyl)phenyl]methyl}-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
N-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-1-(pyrrolidine-1-carbonyl)piperidin-4-amine
N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-4-[(2-methylprop-2-en-1-yl)oxy]benzamide
8-[(2S)-2-amino-3-hydroxypropanoyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-{1'-[2-(azepan-1-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
N-[1-(4-chlorophenyl)cyclobutyl]-2-(2-oxopiperidin-1-yl)acetamide
4-(4-{[2-(1H-indol-1-yl)ethyl]amino}piperidin-1-yl)-N,N-dimethylbenzamide
4-{[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]methyl}pyridine