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N3-cycloheptyl-1-cyclopropyl-N5-[2-(3-fluorophenyl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
methyl[(1-{[1-(6-methylpyridine-3-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]amine
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2-(dimethyl-1,3-thiazol-5-yl)acetamide
(1R,2R,6S,7S)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-10-oxa-4-azatricyclo[5.2.1.02,6]decane
1-[1-(2,4-dimethylphenyl)propyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
2-benzyl-N,1-dimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-5-propanamido-1H-1,3-benzodiazole-7-carboxamide
2-(2-aminoethyl)-N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)quinazolin-4-amine
2-[5-(2-chloro-4-fluorophenyl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-1-yl]acetic acid
N-methyl-3-{[methyl({[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}pyridin-2-amine
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-4-methyl-2-(propan-2-yl)pyrimidine-5-carboxamide
2-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine-4-carbonitrile
N-{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}-N-methyloxan-4-amine
methyl({4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
1-(2-fluoroethyl)-5-(2-methylprop-1-en-1-yl)-4-phenyl-1H-imidazole
N-(2-methylpropyl)-2-(morpholin-4-yl)-N-(thiophen-3-ylmethyl)pyrimidine-5-carboxamide
1-(2-oxopiperidine-3-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-(3-hydroxy-3-phenylpropyl)-N,1-dimethyl-1H-indole-6-carboxamide
2-[methyl(pyridin-2-ylmethyl)amino]-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
6-methoxy-4-[4-(pyridin-3-yl)piperazine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
3-[(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)methyl]-1,2-dihydroquinolin-2-one
5-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)-2-methyl-1,4-dihydropyridin-4-one
1-(4-{[5-(methoxymethyl)furan-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-2,2-diphenylethan-1-ol
1-(furan-2-ylmethyl)-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}piperidine-3-carboxamide
4-(hydroxymethyl)-1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-ol
8-fluoro-2-({4-[(3-methylphenyl)methyl]piperazin-1-yl}methyl)quinoline
2-(2,3-difluorophenyl)-2-[methyl(oxan-4-ylmethyl)amino]acetic acid
8-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
8-[(3-fluorophenyl)methyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[(1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-3-yl)methyl]pyridine-3-carboxamide
5-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}-3-propyl-1H-pyrazole
(4aR,7aS)-1-(2-methylpropanoyl)-4-(1H-pyrrole-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4S)-N-ethyl-1-[(2-fluoro-4-methoxyphenyl)methyl]-4-propanamidopyrrolidine-2-carboxamide
3-ethyl-2-[3-(pyridin-3-ylmethyl)piperidine-1-carbonyl]-1H-indole
{1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-4-[(4-methoxyphenyl)methyl]piperidin-4-yl}methanol
3,5-dichloro-N,4-dimethyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}benzamide
1-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-5-(oxolan-3-yl)-4-phenyl-1H-imidazole
N,6-dimethyl-N-[3-(1H-pyrazol-1-yl)propyl]-2-(pyridin-3-yl)pyrimidin-4-amine
7-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-4-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(2,4-dichlorophenoxy)-1-[(3S,4S)-3-hydroxy-4-(propan-2-yloxy)pyrrolidin-1-yl]ethan-1-one
2-(3-fluoro-4-hydroxyphenyl)-1-{2-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}ethan-1-one
2-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-5-(dimethylamino)-2,3-dihydropyridazin-3-one
2-(2,3-dihydro-1H-inden-1-yl)-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
1-(4-hydroxy-4-phenylpiperidin-1-yl)-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
N,1-dimethyl-N-[2-phenyl-1-(1-{[4-(pyrrolidin-1-yl)phenyl]methyl}piperidin-4-yl)ethyl]-1H-pyrazole-3-carboxamide
4-chloro-1-methyl-3-{[4-(thian-4-yl)piperazin-1-yl]methyl}-1H-indazole
2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
4-({2-[1-(1-ethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
1-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-(pyridin-2-ylmethyl)-1,4-diazepane