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N-methyl-N-(2-methylpropyl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
N-[(3S,7S,8aS)-1,4-dioxo-3-propyl-octahydropyrrolo[1,2-a]piperazin-7-yl]benzamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-5-methylpiperidin-2-one
1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(4-hydroxypiperidin-1-yl)ethan-1-one
N-(1-benzothiophen-5-ylmethyl)-2-(pyrrolidin-3-yl)acetamide
(3R,9aR)-8-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
8-(1-methyl-1H-pyrazole-5-carbonyl)-2-(2-methylpropyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-N,N-diethylpyrrolidin-3-amine
N-{3-[6-amino-5-cyano-4-(4-hydroxy-3-methoxyphenyl)pyridin-2-yl]phenyl}acetamide
6-methyl-2-(2-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)-3,4-dihydropyrimidin-4-one
4-{[6-(2-fluoro-3-methylphenyl)pyridin-3-yl]methyl}morpholine
N-methyl-5-(propan-2-yl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
2-(ethylamino)-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidine-5-carboxamide
N-ethyl-8-methyl-2-(2-methylpyrimidin-5-yl)-N-(pyridin-2-ylmethyl)quinoline-4-carboxamide
3-{[(1-hydroxycyclohexyl)methyl]carbamoyl}-5-methoxybenzoic acid
2-methoxy-N-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
(1R,2S)-1-{4-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]-1H-1,2,3-triazol-1-yl}-2,3-dihydro-1H-inden-2-ol
methyl 3-[({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)carbamoyl]propanoate
3-{2-methyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}propanamide
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-(4-methyl-1,3-oxazole-5-carbonyl)piperidine
7-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-N,N,2-trimethyl-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
(3S,5R)-N3-cyclopentyl-N5-(2,3-dihydro-1H-inden-5-yl)-1-[(4-hydroxyphenyl)methyl]piperidine-3,5-dicarboxamide
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
4-methoxy-N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]benzamide
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-2-(1H-1,2,4-triazol-1-yl)acetamide
1-[1'-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
methyl 1-[(3S,5S)-1-benzyl-5-{[(4-methoxyphenyl)methyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
3-methyl-6-(3-methyl-3-phenylpiperidin-1-yl)pyridazine
N-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-4-yl}-2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidine-1-carboxamide
methyl 7-oxo-3-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]-9-(propan-2-yloxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(dimethylamino)-N-[5-({ethyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]carbamoyl}amino)-2-methylphenyl]acetamide
1-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-3-{imidazo[1,2-a]pyridin-2-yl}propan-1-one
N-[4-(ethylcarbamoyl)-2-methylphenyl]-2-(1,3-thiazol-2-yl)pyrrolidine-1-carboxamide
1-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(pyridin-3-yl)ethane-1,2-dione
1-(1-ethyl-1H-pyrazole-5-carbonyl)-4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
1-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-indazole-3-carboxylic acid
5,8-dimethyl-2-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}quinolin-4-ol
1-benzyl-4-[3-(pyrazin-2-yl)propanoyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
N-{2-[2-(1H-imidazol-2-yl)-1H-imidazol-1-yl]ethyl}-4-methylpyridin-2-amine
3-[({1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}oxy)methyl]pyridine
4-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-3-phenyl-1,2-oxazole
(2S,4S)-4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxylic acid
(2R,3S,6R)-3-(2-methoxyphenyl)-5-[2-(1H-pyrazol-4-yl)ethyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
4-hydroxy-1-methyl-N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)piperidine-4-carboxamide
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-(2-oxopyrrolidin-1-yl)propanamide
1-[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(methylamino)ethan-1-one
2-cyclopropyl-8-[(4-fluorophenyl)methanesulfonyl]-2,8-diazaspiro[5.5]undecan-3-one
N-cyclobutyl-5-{1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
2-(2-fluoro-5-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine