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5-methyl-N-{4-[2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetamido]phenyl}furan-2-carboxamide
3-{7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}-2H-chromen-2-one
N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-2-methylpyrido[2,3-d]pyrimidin-4-amine
4-(1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}azetidin-3-yl)morpholine
4-{1-butyl-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl}pyridine
2-[(1-methylpiperidin-4-yl)(pyridin-3-ylmethyl)amino]-N-(pyridin-2-ylmethyl)acetamide
6-[4-(furan-3-ylmethyl)piperazin-1-yl]-9H-purine
2-(1H-1,3-benzodiazol-1-yl)-1-[3-(2-methoxybenzoyl)piperidin-1-yl]ethan-1-one
N,N-diethyl-1-[(1s,4s)-4-{[(3-ethoxy-2-hydroxyphenyl)methyl]amino}cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-[4-({4-[(3S,4R)-4-hydroxyoxolan-3-yl]-1,4-diazepan-1-yl}methyl)phenoxy]acetic acid
2-ethyl-N,N-dimethyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-4-(thian-4-yl)piperazine
[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)[(2,4,5-trimethoxyphenyl)methyl]amine
N-[(2S,4R,6R)-2-[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]-6-(propan-2-yl)oxan-4-yl]acetamide
1-[4-(1,3-benzoxazol-2-yl)piperidin-1-yl]-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-ethyl-8-[(5-methylpyrazin-2-yl)methyl]-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
2-methoxy-4-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
{[5,8-dimethoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
1-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-5-(4,4,4-trifluorobutan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-{1-[3-(dimethylamino)-2,2-dimethylpropyl]-4-phenyl-1H-imidazol-5-yl}phenol
methyl 2-[5-(8-hydroxyquinolin-2-yl)-4-phenyl-1H-imidazol-1-yl]acetate
5-(2,4-difluorophenoxymethyl)-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
2-{3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-3,4-dihydroquinazolin-4-one
3-[5-(2-methyl-1,3-thiazole-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-N-(propan-2-yl)propanamide
2-(5-ethyl-1-benzofuran-3-yl)-N-[(1-methylpyrrolidin-3-yl)methyl]acetamide
1-{5-benzyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}azetidin-3-ol
2-methyl-7-(3-methyl-1H-pyrazole-5-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(2H-1,3-benzodioxol-5-yl)-2-(morpholin-4-yl)acetic acid
1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-3-(2-methylphenoxy)azetidine
5-[4-(piperidine-1-carbonyl)pyridin-2-yl]pyrimidine
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-1-(3-phenylpropyl)piperidin-3-amine
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)({imidazo[1,2-a]pyrimidin-2-ylmethyl})amine
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(oxan-4-yl)piperidine
methyl 4-[4-(5-cyclopropyl-1,3-oxazole-4-carbonyl)piperazin-1-yl]benzoate
2-amino-6-ethyl-4-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
6-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyrazine-2-carboxamide
(3R,4S)-4-(4-methoxyphenyl)-1-(1H-pyrrole-2-carbonyl)pyrrolidin-3-amine
6-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidin-4-amine
(3aR,6aS)-5-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)-1-oxo-2-propyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[4-(1H-pyrazol-1-yl)phenyl]-1-(thiophen-3-ylmethyl)piperidine-2-carboxamide
2-(4-methyl-1H-imidazol-5-yl)-1-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-1H-imidazole
1-(4-{5-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-2-methoxyphenoxy}piperidin-1-yl)ethan-1-one
(4S)-4-(propan-2-yl)-3-[(2,3,5,6-tetrafluoro-4-methoxyphenyl)methyl]-1,3-oxazolidin-2-one
1-[(2,3-difluorophenyl)methyl]-4-[1-(furan-3-carbonyl)pyrrolidin-3-yl]piperidine
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
6-[2-(2-phenyl-1,3-thiazol-4-yl)acetyl]-N-[4-(1H-pyrazol-1-yl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
4-{5-[2-(2-phenylethyl)piperidine-1-carbonyl]pyrimidin-2-yl}morpholine
2-butoxy-1-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
ethyl 4-(3-phenylpropyl)-1-[2-(pyrimidin-2-ylsulfanyl)acetyl]piperidine-4-carboxylate