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N-methyl-3-(1-methyl-1H-pyrrol-2-yl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1H-pyrazole-5-carboxamide
6-{1-[4-(pyridin-2-yl)pyrimidin-2-yl]piperidin-3-yl}pyrimidin-4-ol
1-{1-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}-N-cyclopropylpiperidine-4-carboxamide
4-(4-methoxyphenoxy)-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
(3aS,7aR)-5-methyl-2-[2-(1H-pyrazol-1-yl)benzoyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
1-[(3S,4S)-3,4-dihydroxypiperidin-1-yl]-2-methyl-2-[5-methyl-2-(propan-2-yl)phenoxy]propan-1-one
2-(2-methoxyphenyl)-N-(1-methyl-1H-pyrazol-5-yl)pyrrolidine-1-carboxamide
2-(4-chlorophenyl)-4-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}morpholine
3-(benzylsulfanyl)-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}propan-1-one
2-(5-tert-butyl-1H-pyrazol-3-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-[6-(2-aminoethyl)-2-methylpyrimidin-4-yl]-1λ6-thiomorpholine-1,1-dione
N-[1-(1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopentanecarboxamide
N-[4-({1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}sulfamoyl)phenyl]acetamide
8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(2-methylpropyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(4-methylpyrimidin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
methyl 4-{[4-(4-fluorophenyl)-1,4-diazepan-1-yl]methyl}-1H-pyrazole-3-carboxylate
N-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[6-oxo-4-(piperazin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
2-{[2-(2H-1,2,3-benzotriazol-2-yl)acetamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-N-methylpyrimidin-2-amine
3-methyl-8-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-ethyl-N-methyl-N-[4-(morpholin-4-yl)butyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-(1H-1,3-benzodiazol-2-ylmethyl)-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]piperidine-3-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-5-hydroxypyrazine-2-carboxamide
8-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[phenyl(pyridin-4-yl)methyl]-1-(propan-2-yl)-1H-pyrazole-3-carboxamide
3-[1-(6-cyclopropylpyrimidin-4-yl)piperidin-4-yl]benzonitrile
2-methyl-3-{[4-(1H-pyrazol-3-yl)piperidin-1-yl]methyl}quinoxaline
6-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[(5-propylfuran-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-methoxy-N-({1-[2-(pyridin-2-yl)acetyl]piperidin-3-yl}methyl)benzene-1-sulfonamide
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-N-[2-(thiophen-2-yl)ethyl]-1H-pyrazole-4-carboxamide
N1,N1-dimethyl-N4-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)piperidine-1,4-dicarboxamide
N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)imidazo[1,2-a]pyridine-6-carboxamide
(3S,4S)-1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-4-propylpyrrolidine-3-carboxylic acid
1-(3-{4-[hydroxy(pyridin-2-yl)methyl]piperidin-1-yl}-3-oxopropyl)-4,6-dimethyl-1,2-dihydropyrimidin-2-one
2-methoxy-N-[2-methoxy-5-({[2-(1,3-thiazol-4-yl)ethyl]carbamoyl}amino)phenyl]acetamide
2-{1-[(4-ethoxyphenyl)methyl]-4-(pyridin-2-ylmethyl)piperazin-2-yl}ethan-1-ol
N-{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-N-methyloxan-4-amine
N-[2-(3-propoxyphenyl)ethyl]-1,9-dioxaspiro[5.5]undecan-4-amine
2-(1-ethylpiperidin-4-yl)-1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}ethan-1-one
4-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1-(4-methoxyphenyl)pyrrolidin-2-one
1-(cyclopropylmethyl)-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
2-(2,5-dimethoxyphenyl)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methylacetamide
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]benzamide
5-(4-methylpiperazine-1-carbonyl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-2-one
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-5-(hydroxymethyl)furan-2-carboxamide
2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-(2-phenylpropan-2-yl)acetamide