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(2R)-2-[({4-[2-(dimethylamino)ethoxy]phenyl}methyl)amino]propanamide
5-(cyclohexylamino)-1-(3-methylbutyl)azepan-2-one
1-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}urea
1-benzoyl-N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-amine
3-benzyl-8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[1,3-dioxo-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidine-4-carboxamide
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl]methanol
methyl (2S,4R)-1-[3-(cycloheptylcarbamoyl)propanoyl]-4-hydroxypyrrolidine-2-carboxylate
2-(methoxymethyl)-3-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-6-methyl-1-(3-phenylpropyl)-1,4-dihydropyridin-4-one
1-(2-methoxyethyl)-8-methyl-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
3-(4-{[3-(5-methylfuran-2-yl)phenyl]methyl}piperazin-1-yl)-1,2-dihydropyrazin-2-one
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(1,2-oxazol-3-ylmethyl)acetamide
benzyl 4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
1-(furan-2-ylmethyl)-4-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}piperidine
2-cyclopropyl-4-methyl-N-[2-(pyridin-2-ylsulfanyl)ethyl]pyrimidine-5-carboxamide
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(4aR,7aS)-1-ethyl-4-(2-fluoro-6-methoxybenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
9-(2,5-dimethylfuran-3-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-cyclopropyl-5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]pyrimidine
3-({[(2,6-difluoro-3-methoxyphenyl)methyl]amino}methyl)pyrrolidin-3-ol
2-(cyclopropylmethyl)-N-(4-ethylphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
[(3-{[1-(3-fluorobenzoyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(2-phenylethyl)amine
6-methyl-N-[(2-phenoxypyridin-3-yl)methyl]pyridine-3-carboxamide
4-[(2,6-dimethylphenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
1-[3-(2-methoxyphenoxy)propyl]-4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridine
2-(3-chloro-4-fluorophenyl)-2-[(3-methyl-1-propyl-1H-pyrazol-4-yl)formamido]acetic acid
5-fluoro-2-{1-[3-(2-methyl-1H-imidazol-1-yl)propyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
2-(4-{[3-(methylsulfanyl)phenyl]methyl}morpholin-3-yl)acetic acid
[(3R,5R)-5-(morpholin-4-ylmethyl)-1-[6-(propan-2-yl)pyridazin-3-yl]piperidin-3-yl]methanol
5-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]-1,2-oxazole-3-carboxamide
1-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]piperidine
[(6-chloroquinolin-2-yl)methyl](methyl)(pyrazin-2-ylmethyl)amine
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(9-ethyl-9H-carbazol-3-yl)methyl]amino}-N-[2-(2-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
methyl 6-{[3-(4-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyridine-2-carboxylate
N-(6-cyanopyridin-3-yl)-2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}morpholine-4-carboxamide
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-(oxolan-2-ylmethoxy)-4-(thiophen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1R,3S)-7-[3-(4-fluorophenyl)benzoyl]-7-azaspiro[3.5]nonane-1,3-diol
1-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-3-(6-methoxy-2H-1,3-benzodioxol-5-yl)urea
2-[1-(ethoxymethyl)cyclobutyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(1S,5R)-3-benzyl-6-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(pyrrolidin-1-yl)ethan-1-one
4-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-5-methyl-1-propyl-1H-pyrazole
1-(2-ethylphenyl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}urea
6-(3-methoxypiperidin-1-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
8-[4-methyl-7-(methylsulfanyl)quinolin-2-yl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
[5-(3-chloro-4-methoxyphenyl)-1H-1,3-benzodiazol-2-yl]methanol
ethyl 1-(oxan-4-yl)-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-1,8-naphthyridine-2-carboxamide