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8-[(2-phenylethyl)carbamoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-[2-({4-benzyl-5-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}sulfanyl)ethyl]morpholine
2-(2H-1,3-benzodioxol-5-yl)-1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
8-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-{5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,4-oxazepane
2-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-3-(piperidine-1-carbonyl)pyrazine
2-(1-methyl-4-{[2-(2-phenylethynyl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-4-(dimethylamino)butanamide
5-(4-acetylphenoxymethyl)-N-cyclopentyl-1,2-oxazole-3-carboxamide
2-[(4-chlorophenyl)methyl]-8-(1H-pyrazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-(2-methoxyethyl)-9-(quinolin-5-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-amino-4-methyl-N-[2-(4-methylmorpholin-2-yl)ethyl]-1,3-benzothiazole-6-carboxamide
1-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-N-methylpyrrolidine-3-carboxamide
1-(2-phenylpropyl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-[4-(1H-imidazol-4-yl)phenyl]-3-[2-(morpholin-4-yl)ethyl]urea
5-[({[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
2-{1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]pyrrolidin-2-yl}-1,3-thiazole
2-[(5-methylpyrazin-2-yl)methyl]-8-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-{[(3aR,6aR)-2-acetyl-octahydropyrrolo[3,4-c]pyrrol-3a-yl]formamido}-N-(1,3-thiazol-2-yl)propanamide
1-{1-[(3-chloro-5-fluorophenyl)methyl]piperidin-4-yl}piperidin-4-ol
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
{1-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methanol
1-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}-N-(2-phenylethyl)piperidine-4-carboxamide
4-[({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]-1-cyclopropylpyrrolidin-2-one
(1S,5R)-3-(3-chloro-4-methylbenzoyl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[2-(azocan-1-yl)-2-oxoethyl]-4-(thiophen-2-ylmethyl)piperazin-2-one
2-[(4aS,8aR)-1-(3-aminopropyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]-N,N-dimethylpyridine-3-carboxamide
2,6-difluoro-3-methoxy-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]benzamide
2-(pyridin-3-yl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]pyrimidine-5-carboxamide
6-cyano-N-methyl-N-[(3-methylthiophen-2-yl)methyl]pyridine-3-carboxamide
(3S)-N,N-dimethyl-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}azepan-3-amine
(1R,5S)-6-(1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carbonyl)-6-azabicyclo[3.2.1]octane
N,N-dimethyl-1-{5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidin-3-amine
2-[(2-{[2-(dimethylamino)ethyl][(5-methylthiophen-2-yl)methyl]carbamoyl}phenyl)amino]acetic acid
1-[7-(3-chlorophenyl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(thiophen-3-yl)ethan-1-one
(1R,9S)-5-amino-3-[4-(dimethylamino)phenyl]-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
N-[1-(4-methoxyphenyl)ethyl]-N,2,3-trimethyl-1H-indole-7-carboxamide
N-[3-(2-ethoxyphenyl)propyl]-2,3-dimethylquinoxaline-6-carboxamide
2-[3-(oxolan-3-yl)-5-[2-(4H-1,2,4-triazol-4-yl)phenyl]-1H-1,2,4-triazol-1-yl]acetic acid
N-[2-(pyrazin-2-yl)ethyl]-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
1-(3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-4-(morpholin-4-yl)phenyl)ethan-1-one
N,N-dimethyl-5-({2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)pyridin-2-amine
N-butyl-N-[(4-fluorophenyl)methyl]-5-methyl-1,3-oxazole-4-carboxamide
1-[1-ethyl-3-(hydroxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one
N-[2-(diethylamino)ethyl]-N-ethyl-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(2,3-dimethyl-1H-indole-5-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
8-[2-(3-fluorophenyl)acetyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(methylamino)ethyl]-1-[3-(2-methylpyrimidin-4-yl)phenyl]piperidin-4-amine