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N-[(1-{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)methyl]acetamide
(1R,5S,6S)-6-{[4-(diphenylmethyl)piperazin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane
N-[4-({[3-(4-methylphenyl)propyl]carbamoyl}methoxy)phenyl]propanamide
9-[4-(1H-imidazol-1-yl)benzoyl]-5-methoxy-1-oxa-9-azaspiro[5.5]undecane
1-cyclopropyl-N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-5-oxopyrrolidine-3-carboxamide
3-(propan-2-yl)-5-[(2S)-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]pyrrolidin-2-yl]-1,2,4-oxadiazole
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]-N-propylacetamide
N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-[4-(difluoromethoxy)benzoyl]-3-(3-methoxypropyl)piperidine
3-{2-[4-(2-methoxyethoxy)piperidin-1-yl]-2-oxoethyl}-4-(3-methylbutyl)piperazin-2-one
(3R)-1-[6-(azepan-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]pyrrolidin-3-ol
3-(1-benzyl-3-methyl-1H-pyrazol-5-yl)-1-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]urea
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-1-methylcyclopropane-1-carboxamide
methyl (2S,4R)-4-[4-(2,4-dioxoimidazolidin-1-yl)benzamido]-1-methylpyrrolidine-2-carboxylate
2-methoxy-1-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-phenylethan-1-one
3-[(3R,4S)-1-{6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
2-[4-(cyclopropylmethyl)piperazine-1-carbonyl]-N,N-dimethyl-2,3-dihydro-1H-inden-2-amine
5-oxo-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
2-(1H-1,3-benzodiazol-2-yl)-1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl]methanol
N-[4-(ethylsulfanyl)phenyl]-3-(pyridine-2-carbonyl)piperidine-1-carboxamide
3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}-N-(furan-2-ylmethyl)piperidine-1-carboxamide
methyl 3-[(3S,4R)-1-[(2,4-dimethoxy-3-methylphenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoate
(2E)-3-(3-fluorophenyl)-N-(oxolan-2-ylmethyl)-N-{[3-(thiophen-3-ylmethoxy)phenyl]methyl}prop-2-enamide
1-[2-(dimethylamino)ethyl]-5-oxo-N-[2-(pyridin-3-yl)ethyl]pyrrolidine-3-carboxamide
3-{1-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1H-imidazol-2-yl}-1,2-dihydroquinolin-2-one
ethyl 4-[({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]piperidine-1-carboxylate
4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-2-(trifluoromethyl)morpholine
7-methoxy-N-[3-(4H-1,2,4-triazol-4-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-ethyl-1-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(5-methylfuran-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[2-(propan-2-yloxy)ethyl]-1,3-oxazole-4-carboxamide
3-[5-(1-benzofuran-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-N-(2-hydroxyethyl)propanamide
(3R,4R)-1-[4-(3-fluorophenyl)benzoyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
{6-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]pyridin-2-yl}methanol
5-[3-methyl-4-(morpholin-4-yl)benzoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
2-{3,5-dimethyl-4-[2-(pyridin-4-yl)-1H-imidazol-1-yl]-1H-pyrazol-1-yl}ethan-1-ol
4-(4-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl](methyl)amino}piperidin-1-yl)-N-[2-(morpholin-4-yl)ethyl]benzamide
(1R,5S,8S)-N-(3-cyclopentaneamidophenyl)-8-methoxy-3-azabicyclo[3.2.1]octane-3-carboxamide
(2R,3R)-3-[4-(2-methoxyphenyl)-1H-1,2,3-triazol-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-{2-[4-hydroxy-4-(pyridin-2-yl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylic acid
(1s,4s)-N-({1-[(3,5-dimethylphenyl)methyl]pyrrolidin-3-yl}methyl)-4-hydroxycyclohexane-1-carboxamide
1-benzyl-5-methyl-4-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-1H-1,2,3-triazole
(1S,5R)-6-(dimethyl-1,2-oxazole-4-carbonyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-{1-[4-(3-chlorophenyl)-5-({[3-(trifluoromethyl)phenyl]methyl}sulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}-4-methoxybenzamide
2-benzyl-8-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
(3R,4R)-1-[1-(2,3-dihydro-1H-inden-5-yl)piperidin-4-yl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
N-cyclopropyl-1-(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
N-(1H-1,3-benzodiazol-2-yl)-2-{[cyclopropyl(3-methylpyridin-2-yl)methyl]amino}acetamide