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4-chloro-N-[3-(cyclohexyloxy)propyl]-1-methyl-1H-pyrazole-5-carboxamide
1-[(2-fluorophenyl)methyl]-3-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-N-(pyridin-4-ylmethyl)thiophene-2-carboxamide
(5S)-5-[({[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}(pyridin-2-ylmethyl)amino)methyl]pyrrolidin-2-one
2-[4-(4-amino-3-methoxypyridin-2-yl)phenyl]-2-methylpropanenitrile
7-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-[(2E)-2-methylbut-2-en-1-yl]-2,7-diazaspiro[4.5]decane
3-(1H-1,2,3-benzotriazol-4-yl)-1-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]urea
2-ethyl-4-phenyl-9-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-2,9-diazaspiro[5.5]undecane
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)propanamide
4-[4-(1-ethoxyethyl)phenyl]-6-methyl-2,3-dihydropyridazin-3-one
(1R,6S)-N-(dimethyl-1,2-oxazol-4-yl)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
1-(1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)-4-(2-methoxyethyl)piperazine
2-(furan-2-yl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-benzyl-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-({[4-(methylsulfanyl)phenyl]methyl}(propyl)amino)propane-1,2-diol
N-[(3-fluorophenyl)methyl]-9-methoxy-3-[2-(methylsulfanyl)benzoyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[2-(4-fluorophenoxy)ethyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
9-(3-hydroxy-4-methoxybenzoyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(2,2,2-trifluoroethyl)acetamide
2-[(5-ethylpyridin-2-yl)methyl]-2,7-diazaspiro[4.5]decane
N-[4-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-6-hydroxy-1,4-oxazepane-4-carboxamide
3-methyl-6-[5-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-3-yl]pyridazine
4-fluoro-N-(2-{[3-(piperidin-3-yl)phenyl]formamido}ethyl)benzamide
N-[1-(4-fluorophenyl)piperidin-4-yl]-2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]acetamide
N,N,4-trimethyl-5-(thiomorpholine-4-carbonyl)pyrimidin-2-amine
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
1-{3-[4-({[2-(cyclohex-1-en-1-yl)ethyl]amino}methyl)-2-methoxyphenoxy]-2-hydroxypropyl}piperidin-4-ol
(3S,5R)-1-benzyl-N3-[3-(dimethylamino)propyl]-N5-(4-fluorophenyl)piperidine-3,5-dicarboxamide
(2R)-2-[4-phenyl-5-(quinolin-3-yl)-1H-imidazol-1-yl]propanamide
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-2,2-dimethylpropan-1-one
3-benzyl-4-(quinoxaline-6-carbonyl)piperazin-2-one
3-methyl-5-[({[3-(2-methylpropyl)-1-phenyl-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)methyl]-1,2,4-oxadiazole
(3S,5R,9R)-5-hydroxy-11-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(3-methoxy-2-methylbenzoyl)pyrrolidin-3-yl]methanol
2-methyl-4-[4-(5,6,7,8-tetrahydro-1,6-naphthyridine-6-carbonyl)phenyl]butan-2-ol
3-(3-hydroxybutyl)-6-methyl-3,4-dihydroquinazolin-4-one
4-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1-methyl-1,2-dihydroquinolin-2-one
1-benzyl-N-methyl-N-(pyrimidin-4-ylmethyl)-1H-pyrazole-4-carboxamide
{[4-ethyl-5-(1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl}dimethylamine
1-(5-methoxy-2-methylphenyl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
1-ethyl-4-[4-(pyridin-4-ylmethyl)piperazine-1-carbonyl]pyrrolidin-2-one
3-({4-[4-(3-methoxyphenyl)-5-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}acetamide
1-{2-[(3-methylpyridin-2-yl)amino]ethyl}-3-(1,3,6-trimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(oxan-4-yl)piperidine
[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]({[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl})amine
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(4-methoxy-2-methylphenyl)methyl]piperidine
3-({[(3-hydroxyphenyl)methyl](methyl)amino}methyl)-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
3,3-dimethyl-1-[(5-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]urea