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N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-2-(ethylamino)pyrimidine-5-carboxamide
1-(furan-2-carbonyl)-4-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}-1,4-diazepane
2-methoxy-N-(1-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]butanamide
2-amino-6-(1-methyl-1H-pyrrol-3-yl)-4-[5-(oxan-2-yl)furan-2-yl]pyridine-3-carbonitrile
[4-(1-cyclopropanecarbonylpiperidine-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methanol
methyl 1-[(3R,5S)-1-[(3-methoxyphenyl)methyl]-5-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-N-(1,3-thiazol-2-ylmethyl)cyclopropanamine
2-[(4-methyl-1H-1,3-benzodiazol-2-yl)methoxy]-N-[(1-methylpiperidin-3-yl)methyl]acetamide
[(2-fluorophenyl)methyl]({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl})amine
1-(cyclohexylmethyl)-N-[(6-hydroxypyrimidin-4-yl)methyl]-6-oxopiperidine-3-carboxamide
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-[3-(thiophen-2-yl)propanoyl]piperidine-2-carboxamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-(5-phenyl-1,2-oxazole-3-carbonyl)piperazine
2-[1-(2,3-dihydro-1H-inden-2-yl)-5-[(2S)-1-propanoylpyrrolidin-2-yl]-1H-1,2,4-triazol-3-yl]acetamide
3-[(3S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-1-(4-hydroxypiperidin-1-yl)propan-1-one
4-fluoro-1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidine
5-[(1S,5S)-3,6-diazabicyclo[3.2.2]nonan-3-ylmethyl]-N,N-dimethylpyridin-2-amine
4-ethyl-5-methyl-6-[4-(pyrazin-2-yl)piperazin-1-yl]pyrimidin-2-amine
5-[(6,7-dimethoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
4-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-methyl-5-({1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}methyl)furan-2-carboxamide
(2R)-N-[1-(4-fluorophenyl)-4-(morpholin-4-yl)-1H-indazol-3-yl]oxolane-2-carboxamide
1-cyclopentanecarbonyl-N-methyl-N-(1,2-oxazol-3-ylmethyl)piperidine-4-carboxamide
methyl 5-{[(2E)-4-methylpent-2-en-1-yl]amino}-3-(oxolane-3-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[2-(1H-imidazol-4-yl)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[(2-fluorophenyl)methyl]-3-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-yl}propanamide
3-{[(2-methoxyphenyl)methyl](prop-2-en-1-yl)amino}propane-1,2-diol
methyl 1-[(3S,5S)-1-[1-(2-phenylethyl)piperidin-4-yl]-5-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-[2-(1H-imidazol-4-yl)ethyl]-9-{2-[methyl(propan-2-yl)amino]acetyl}-2,9-diazaspiro[5.5]undecan-3-one
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methylacetamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
7-(5-chloropyridin-2-yl)-4-[(3-fluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethan-1-one
N-benzyl-N-methyl-1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-amine
6,7-dimethoxy-2-(pyridin-3-yl)quinazolin-4-amine
4-[(3-{2-[4-(hydroxymethyl)phenyl]pyridin-4-yl}pyrrolidin-1-yl)methyl]-2-methylphenol
(3S,5R)-N-(4-methylphenyl)-5-[4-(propan-2-yl)piperazine-1-carbonyl]piperidine-3-carboxamide
1-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(3-methylphenyl)ethan-1-one
8-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
ethyl 4-[4-(4-{methyl[2-(oxan-2-yl)ethyl]amino}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
1-(3-chlorophenyl)-4-(1-methyl-1H-pyrrole-2-carbonyl)piperazin-2-one
1-{3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propanoyl}-1,4-diazepane-6-carboxylic acid
N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}pyrazolo[1,5-a]pyridine-3-carboxamide
4-[1-(2-propoxyacetyl)piperidin-3-yl]benzoic acid
N-[(3R,4S)-4-cyclopropyl-1-(2-hydroxyethyl)pyrrolidin-3-yl]pyrazine-2-carboxamide
N3-(1,3-benzothiazol-2-ylmethyl)-N5-benzyl-N3-methyl-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[(3S,4R)-4-(4-methylphenyl)-1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)pyrrolidin-3-yl]acetamide
1-(difluoromethyl)-N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1H-pyrazole-3-carboxamide
5-[3-(3-methylphenyl)piperidine-1-carbonyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidin-4-ol
N-[(2-phenoxypyridin-3-yl)methyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide