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N-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}-2-(4-phenylpiperidin-1-yl)acetamide
4-benzyl-3-ethyl-1-(3-fluoropyridine-4-carbonyl)-1,4-diazepan-5-one
1-{1-[(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-2,3-dihydro-1,2-benzothiazol-3-one
(4-{4-[1-(2-phenylethyl)pyrrolidin-3-yl]pyridin-2-yl}phenyl)methanol
N-[(5-methylpyrazin-2-yl)methyl]-2-(pyrrolidin-3-yl)benzamide
1-(4-{[2-(1H-imidazol-4-yl)ethyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
6-{4-[1-(dimethylamino)ethyl]phenyl}-N-(propan-2-yl)pyridazin-3-amine
2,5-dimethyl-7-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-[1,3]oxazolo[5,4-d]pyrimidine
(3aS,6aS)-2-[(4-acetylphenyl)carbamoyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(2-benzyl-1,3-benzoxazole-5-carbonyl)piperidine-3-carboxamide
3-{1-[2-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-2-yl}pyridine
4-(benzyloxy)-1-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidine
2-methyl-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}imidazo[1,2-a]pyridine-3-carboxamide
4-(2-{4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]morpholin-3-yl}acetyl)piperazin-2-one
3-[ethyl(oxan-4-ylmethyl)amino]-1-(3-methylpiperidin-1-yl)propan-1-one
7-(5-chloropyridin-2-yl)-4-cyclobutanecarbonyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
7,7-dimethyl-N-[(5-methylfuran-2-yl)methyl]-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
methyl 2-[(3,5-dimethylphenyl)sulfamoyl]-6-(4-methylpentanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-(2-chloro-4-methoxyphenoxymethyl)-N-(pentan-3-yl)-1H-pyrazole-3-carboxamide
(3R,4R)-1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
8-fluoro-2-(morpholin-4-ylmethyl)quinolin-4-ol
N-(3-methoxypropyl)-N-{[6-(thiophen-2-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}oxolane-2-carboxamide
1-(3-chloro-4-methoxybenzoyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
N-[(5-ethylfuran-2-yl)methyl]-4-methyl-5-{1-[2-(morpholin-4-yl)ethyl]-1H-pyrazol-3-yl}-1,3-thiazol-2-amine
N-methyl-N-[2-(2-methylphenyl)-1-{1-[2-(phenylsulfanyl)acetyl]piperidin-4-yl}ethyl]cyclobutanecarboxamide
3-{[2-({3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1H-pyrrol-1-yl]methyl}pyridine
(3R,4R)-1-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-4-ethylpiperidine-3,4-diol
1-butyl-3-[2-(methylsulfanyl)ethyl]-5-(pyrrolidin-1-ylmethyl)-1H-1,2,4-triazole
5-{3-[2-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-oxopropyl}-5-(thiophen-2-ylmethyl)pyrrolidin-2-one
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
1-(2,3-dihydro-1H-inden-2-yl)-4-[(1H-imidazol-4-ylmethyl)amino]pyrrolidin-2-one
3-(1-{[4-(2-hydroxyethoxy)phenyl]methyl}piperidin-3-yl)-N-[4-(trifluoromethyl)phenyl]propanamide
3-[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraene
4-cyclopropyl-6-[4-(2-methoxyphenyl)piperidin-1-yl]pyrimidine
3-[1-(5-ethyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
3-[1-({5-[1-(2-methoxyethyl)-1H-pyrazol-3-yl]thiophen-2-yl}methyl)piperidin-2-yl]pyridine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(2-oxopyrrolidin-1-yl)acetamide
N-[2-(dimethylamino)ethyl]-3-[1-(quinolin-2-yl)piperidin-4-yl]propanamide
1-cyclobutanecarbonyl-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]piperidine-4-carboxamide
2-amino-4-(3,5-dimethoxyphenyl)-6-(propan-2-yl)pyridine-3-carbonitrile
5-{2-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-(4-methyl-1H-pyrazol-1-yl)-1-(quinolin-2-ylmethyl)piperidine-4-carboxylic acid
2-fluoro-N-{1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-5-sulfamoylbenzamide
3-(3-fluorophenoxymethyl)-1-(1H-1,2,3-triazole-5-carbonyl)piperidine
2-methyl-6-(1-{[2-(5-methylfuran-2-yl)phenyl]methyl}piperidin-4-yl)-3,4-dihydropyrimidin-4-one
(3S,4R)-1-(5-chloro-1H-indole-2-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl][1-(morpholin-4-yl)propan-2-yl]amine
N-(propan-2-yl)-1-[(1s,4s)-4-[3-(3-methoxyphenyl)propanamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl](1,4-dioxan-2-ylmethyl)methylamine