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5-cyclopropyl-N-(1,4-dioxan-2-ylmethyl)-N-methyl-1,3,4-oxadiazol-2-amine
{3-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]phenyl}methanol
2-[3-(prop-2-en-1-yloxy)benzoyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
7-(4-methyl-1H-pyrrole-2-carbonyl)-N-(oxolan-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-methyl-4-{1-[(3-phenoxyphenyl)methyl]pyrrolidin-3-yl}piperazine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
8-[4-(1H-indol-3-yl)butan-2-yl]-3-[(4-methoxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3aR,6aR)-2-[3-(1H-imidazol-1-yl)propyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl 4-{[4-(4-fluorophenoxy)piperidine-1-carbonyl]amino}benzoate
(3R,4S)-4-cyclopropyl-N,N-dimethyl-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]pyrrolidin-3-amine
N-(3-phenylprop-2-yn-1-yl)-N-(prop-2-en-1-yl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
2-butyl-8-(1-methyl-1H-indole-6-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
8-[(1r,4r)-4-methylcyclohexanecarbonyl]-2,8-diazaspiro[4.5]decan-3-one
2-{5-[(4aR,8aR)-octahydro-2H-1,4-benzoxazin-4-ylmethyl]furan-2-yl}benzonitrile
4-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-6-methoxypyrimidin-2-amine
N-[(3S,4R)-1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
4-{[(5-chloro-2-methoxyphenyl)methyl](methyl)amino}-N-cyclopropylpyridine-2-carboxamide
8-[(5-chlorothiophen-2-yl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(4,6-dimethylpyrimidin-2-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}piperidin-4-amine
2-(1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)-1,3-benzoxazole
4-{6-[(2S)-4-methyl-2-phenylpiperazin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}morpholine
3-[(2R,3R,6R)-5-[(2,4-difluorophenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
(3S,9aR)-3-benzyl-8-(4-methylbenzenesulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(2R)-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}oxolane-2-carboxamide
3-{4-[2-fluoro-3-(trifluoromethyl)phenyl]-1H-pyrazol-1-yl}propanamide
N-[(3S)-2-oxoazepan-3-yl]-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-2-(trifluoromethyl)benzamide
1-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}-3-(piperazin-1-yl)propan-1-one
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-1-methyl-N-(oxolan-2-ylmethyl)piperidin-4-amine
(1R,7S)-N-(1H-imidazol-2-ylmethyl)-3-[(3-methoxyphenyl)methyl]-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
4-{[(1,4-dioxan-2-ylmethyl)carbamoyl]amino}-N-ethyl-N-phenylbenzamide
3-hexyl-8-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-benzyl-1-methyl-8-(3-phenylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-2-carbonitrile
N-[2-(pyridin-2-ylsulfanyl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-({1-[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]propan-2-yl}oxy)pyridine
4-methyl-6-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-2-phenylpyrimidine
methyl (2S,4R)-4-(2,6-dimethylpyrimidine-4-amido)-1-methylpyrrolidine-2-carboxylate
2-{3-[(1-methylpiperidin-4-yl)methyl]-5-[(2-oxo-1,2-dihydropyridin-1-yl)methyl]-1H-1,2,4-triazol-1-yl}acetic acid
4-(1H-imidazol-1-yl)-1-(2-propyl-1,3-thiazole-4-carbonyl)piperidine-4-carboxylic acid
3,3-dimethyl-1-{[5-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}urea
1-(furan-2-ylmethyl)-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]piperidine-4-carboxamide
1-(2,2-dimethylpropyl)-3-hydroxy-3-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)piperidin-2-one
2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-[(3-ethenylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(1S,6R)-9-[5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carbonyl]-3-methyl-3,9-diazabicyclo[4.2.1]nonane
6-fluoro-N-[1-(4-methylpyridin-2-yl)propyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
5-(dimethyl-1,3-oxazol-5-yl)-1-[(4-ethylphenyl)methyl]-1H-1,2,4-triazole
4-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)-1λ6-thiane-1,1-dione
2-(piperidine-1-carbonyl)-6-(2,4,6-trimethylphenyl)pyrazine