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8-[(2-chloro-3,4-dimethoxyphenyl)methyl]-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(4aS,7aR)-1-[2-(2,5-dimethylphenyl)acetyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(methylamino)pyrimidine-5-carboxamide
3-[2-(dimethylamino)ethyl]-1-ethyl-8-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
(1R,7S)-3-(2-methoxyethyl)-N-methyl-N-(1,2-oxazol-5-ylmethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-2,3-dimethylquinoxaline-6-carboxamide
2-hydroxy-5-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}methyl)benzoic acid
2-[(1S,5R)-3-(4-cyclobutyl-6-methylpyrimidin-2-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(propane-1-sulfonyl)-decahydro-1,6-naphthyridin-2-one
(3aS,6aR)-5-(4-fluorobenzoyl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
methyl[(2-methyl-1,3-oxazol-4-yl)methyl][(2-phenyl-1,3-thiazol-4-yl)methyl]amine
1-amino-N-({1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidin-3-yl}methyl)cyclopentane-1-carboxamide
(1R,5S,8S)-3-({3-methoxy-4-[(4-methylphenyl)methoxy]phenyl}methyl)-3-azabicyclo[3.2.1]octan-8-ol
5-{[1-(2-methoxyphenoxy)propan-2-yl]carbamoyl}thiophene-2-carboxylic acid
N-[2-(1H-imidazol-4-yl)ethyl]-1-[4-(4-methylphenyl)phenyl]piperidin-4-amine
3-(3-methyl-3-phenylpiperidin-1-yl)propanoic acid
N-benzyl-N-methyl-1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-3-amine
1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2-methyl-1,4-diazepan-5-one
2-{4-[(2-methyl-1H-imidazol-4-yl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
2-(1-{[1-(1-propylpiperidin-4-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
3-[2-(6-methoxynaphthalen-2-yl)morpholine-4-carbonyl]benzonitrile
3-(2-amino-1,3-thiazol-4-yl)-N-[1-(4-methanesulfonylphenyl)propyl]propanamide
2-methyl-N-[(4-sulfamoylphenyl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
2-(azepan-1-yl)-N-[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethyl]acetamide
(3S,4S)-1-{[4-(cyclopentyloxy)phenyl]methyl}-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
5-(4-hydroxy-1-propylpiperidin-4-yl)-N-methyl-N-(quinolin-8-ylmethyl)-1-benzofuran-2-carboxamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-(1H-imidazol-1-yl)propanamide
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
(3S,4S)-1-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]-4-(piperidin-1-yl)pyrrolidin-3-ol
N-cyclopropyl-N-[(3-ethoxyphenyl)methyl]-2-(pyridin-3-yl)acetamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-{[4-(phenoxymethyl)thiophen-2-yl]methyl}acetamide
N-[2-(1H-indol-3-yl)ethyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
6-{1-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperidin-3-yl}pyrimidin-4-ol
{5-[2-(3-methoxyphenoxy)ethyl]-1H-indol-2-yl}methanol
1-methyl-4-({2-[4-(trifluoromethyl)phenyl]-1H-imidazol-1-yl}methyl)piperidin-4-ol
3-chloro-4-fluoro-N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-benzothiophene-2-carboxamide
1-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-3-methyl-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
6-(4-fluorophenyl)-N-methyl-N-(oxolan-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,2-oxazole-3-carboxamide
(2S)-2-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propanamide
1-[2-(dimethylamino)ethyl]-5-oxo-N-(1,3-thiazol-2-ylmethyl)pyrrolidine-3-carboxamide
N1,N1,N4-trimethyl-N4-{[3-(methylsulfanyl)phenyl]methyl}piperidine-1,4-dicarboxamide
(3aR,5R,6S,7aS)-2-(2,1,3-benzoxadiazol-4-ylmethyl)-octahydro-1H-isoindole-5,6-diol
3-(2,5-dimethoxyphenyl)-5-(1H-pyrazol-4-yl)-1,2,4-oxadiazole
4-(4-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidine-1-carbonyl}piperidin-1-yl)-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
1-{4-[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-2-(2,5-dimethylphenyl)ethan-1-one
3-(6-methoxynaphthalene-2-carbonyl)-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidine
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-2-(1H-pyrazol-1-yl)acetamide