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9-[4-(4-fluorophenyl)benzoyl]-2,9-diazaspiro[5.5]undecan-3-one
4-ethyl-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-1,2,3-thiadiazole-5-carboxamide
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-methyl-2-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidine-1-carbonyl}phenol
ethyl 4-({2-[2-hydroxy-3-(thiomorpholin-4-yl)propoxy]phenyl}methyl)piperazine-1-carboxylate
1-[(1R,5R)-6-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]ethan-1-one
N-(3-methoxyphenyl)-3-{1-[3-(1,2-oxazinan-2-yl)propanoyl]piperidin-4-yl}propanamide
4-[4-(3,5-difluorophenyl)-1H-1,2,3-triazol-1-yl]-1-(thian-4-yl)piperidine
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-3-(prop-2-en-1-yloxy)benzamide
3-(6-methoxypyridin-3-yl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
N,2-dimethyl-N-[(3-methylpyridin-2-yl)methyl]-6-(piperidin-3-yl)pyrimidin-4-amine
6-butyl-2-[4-({methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-3-(thiophen-3-yl)propanamide
N-[(3,5-dimethoxyphenyl)methyl]-3-(1H-pyrazol-4-yl)benzamide
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-[(5-methylfuran-2-yl)methyl]-1,2-oxazole-3-carboxamide
N-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-1-[(2-fluorophenyl)methyl]piperidin-3-amine
(1S,5R)-3-(pyridine-4-carbonyl)-6-(pyrrolidine-1-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
3-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N-methylbenzamide
1-({1-[(1-cyclohexanecarbonylpiperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}methyl)piperazine
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)pyridazine-4-carboxamide
N-[2-(dimethylamino)ethyl]-N-methyl-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-cyclohexyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-methyl-2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
3-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-2-methylphenol
3-(3-hydroxy-3-methylbutyl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
8-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-(3-methyl-1,2,4-oxadiazol-5-yl)-2-[3-(1H-pyrazol-5-yl)piperidin-1-yl]pyridine
5-cyclopropanecarbonyl-1'-(1-methylpiperidine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-[methyl(2-phenylethyl)amino]-N-[3-(methylsulfanyl)phenyl]piperidine-1-carboxamide
1-ethyl-N-[(5-methylfuran-2-yl)methyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
(4S)-3-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-4-(propan-2-yl)-1,3-oxazolidin-2-one
4-(3-methylphenyl)-3-(1H-pyrazol-1-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(ethanesulfonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
methyl (2S,4S)-4-(3,4-dimethoxybenzamido)-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxylate
2-(4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}morpholin-3-yl)-N-(2-methylpropyl)acetamide
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)-1H-pyrazol-1-yl]acetamide
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N-methyl-4-(thiophen-2-yl)butanamide
(2S,4S)-4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetamido]-N-ethyl-1-(1H-imidazol-4-ylmethyl)pyrrolidine-2-carboxamide
N-{1-[1-(1,4-dithiepan-6-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide
5-(2-chloro-4-methoxyphenoxymethyl)-3-[(2R,5S)-2,5-dimethylpyrrolidine-1-carbonyl]-1H-pyrazole
N-(3-cyclohexyl-1H-1,2,4-triazol-5-yl)-3-phenylpiperidine-1-carboxamide
3-(1-methyl-1H-imidazol-2-yl)-6-(naphthalen-1-yl)pyridazine
5-ethyl-N4,6-dimethyl-N4-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrimidine-2,4-diamine
methyl 5-{[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]sulfonyl}-1-methyl-1H-pyrrole-2-carboxylate
1-{furo[3,2-c]pyridin-4-yl}-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
N-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]benzamide
6-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-N4-methylpyrimidine-2,4-diamine
ethyl 4-[3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)propanoyl]piperazine-1-carboxylate