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1-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(methylsulfanyl)ethan-1-one
2-{3-oxo-3-[3-(1H-pyrazol-5-yl)piperidin-1-yl]propyl}-2,3-dihydro-1H-isoindol-1-one
4-(4-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)-1,4-diazepane-1-carbaldehyde
N-[2-(4-methoxyphenyl)ethyl]-N-(pyridin-3-ylmethyl)spiro[2.2]pentane-1-carboxamide
3-(3-methoxyphenyl)-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-pyrazole-5-carboxamide
6-(2-aminoethyl)-N-[3-(phenylsulfanyl)propyl]pyrimidin-4-amine
3-(2-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
2-[(2-methoxybutanamido)methyl]-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
3-{1-[3-(2-chlorophenyl)propanoyl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-(2,4-dioxoimidazolidin-1-yl)-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]benzamide
N-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-1,3-thiazole-5-carboxamide
N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]naphthalene-2-carboxamide
3-{1-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-1H-imidazol-2-yl}phenol
2-methyl-N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]propanamide
9-[3-(1H-pyrazol-1-yl)propanoyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(2-ethylpyrimidin-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(2-methyl-1-benzofuran-7-carbonyl)piperazine
3-[(3R,4S)-1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-4-(dimethylamino)piperidin-3-yl]propanoic acid
1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
1-methyl-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
3-[(4aR,7aS)-4-[(2-methyl-1,3-thiazol-4-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
2-amino-4-(4-fluoro-2-methylphenyl)-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-4-[(1-methylpiperidin-3-yl)methyl]piperazine
1-(2-methoxy-5-{[(2-methoxy-2-methylpropyl)amino]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
1-(2H-1,3-benzodioxol-5-yl)-4-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]piperidine
5-methyl-N-(oxolan-2-ylmethyl)-4-{[(4-phenyloxan-4-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
ethyl 2-[ethyl({[2-(prop-2-en-1-yloxy)phenyl]methyl})amino]acetate
2-(2,6-dimethoxyphenyl)-2-{[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}acetic acid
[2,4,6-trimethyl-3-({[(2S)-3-methylbutan-2-yl]amino}methyl)phenyl]methanol
N-[2-(1H-imidazol-4-yl)ethyl]-3-(1,2-oxazinan-2-yl)propanamide
N-(6-chloro-2-methylpyridin-3-yl)-4-methyl-1,2,3,6-tetrahydropyridine-1-carboxamide
3-methyl-7-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidine-3-carboxamide
1-(2,5-dimethoxybenzoyl)-4-[(3-methylpyridin-2-yl)methyl]piperazine
1-[1-(4-fluorophenyl)-2-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]ethyl]piperidine
N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-2-(4-methylphenyl)quinoline-4-carboxamide
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
N,N-bis(1,3-oxazol-4-ylmethyl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3-(1H-pyrazol-1-ylmethyl)benzamide
2-{7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}acetamide
N-({1-[2-(1H-indazol-3-yl)acetyl]piperidin-3-yl}methyl)-2-(4-methoxyphenyl)acetamide
1-[3-(3-methoxyphenyl)phenyl]-N-(oxan-3-yl)piperidin-4-amine
3-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-4-hydroxy-N-methyl-2-(phenoxymethyl)pyrimidine-5-carboxamide
(3R,4R)-4-methyl-1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-3-(propan-2-yl)pyrrolidin-3-ol
3-(5-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl}-1,2,4-oxadiazol-3-yl)pyridazine
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
5-methyl-N-[1-methyl-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
(4aS,7aR)-1-(3-hydroxypyridine-2-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione