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(3S,4S)-4-[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]-1-(4-methoxybenzoyl)pyrrolidin-3-ol
(2S,4R)-4-amino-1-[(cyclopentylcarbamoyl)carbonyl]-N-ethylpyrrolidine-2-carboxamide
1-(4-{2-[4-(1-hydroxyethyl)piperidin-1-yl]-2-oxoethoxy}phenyl)propan-1-one
N-(2-{3-[2-(4-methoxyphenyl)ethyl]piperidin-1-yl}-2-oxoethyl)methanesulfonamide
3-({[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]amino}methyl)-N-methylbenzamide
N-phenyl-3-{2-[4-(propan-2-yl)morpholin-2-yl]acetamido}propanamide
2-(2,4-dimethoxyphenyl)-6-fluorobenzamide
(1S,4S)-2-(3-chloro-4-methoxyphenyl)-5-(pyridin-2-ylmethyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
2-{[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl](methyl)amino}-N-[(2-methoxyphenyl)methyl]acetamide
2-{1-[3-(pyridin-3-yl)propanoyl]pyrrolidin-3-yl}benzoic acid
4-{1-[1-(5-chloro-2-methylbenzoyl)piperidin-4-yl]ethyl}morpholine
4-{[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
(3S,9aR)-8-(cyclopropylmethyl)-2-methyl-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{1-[(4-ethoxyphenyl)methyl]-4-(1H-indol-2-ylmethyl)piperazin-2-yl}ethan-1-ol
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(2-oxopyrrolidin-1-yl)acetamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(dimethylamino)-N-methyl-2-(2-methylphenyl)acetamide
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carboxamide
4-(3-hydroxy-4-methoxybenzoyl)-1-(3-methoxyphenyl)piperazin-2-one
2-methyl-5-[2-(trifluoromethyl)morpholine-4-carbonyl]phenol
2-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
(2S)-2-amino-4-[3-(carbamoylmethyl)-1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-5-yl]butanoic acid
4-cyclopentyl-N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]pyrimidin-2-amine
3-({[1-(2-methyl-1-benzofuran-5-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-(thiophen-2-ylmethyl)piperazine
1-(2-methyl-4-{methyl[2-(morpholin-4-yl)ethyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)ethan-1-one
N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
N-[(4-methanesulfonylmorpholin-2-yl)methyl]pyrimidin-2-amine
5-(2-{[(3-fluorophenyl)methyl]amino}ethyl)-1-(3-phenylpropyl)pyrrolidin-2-one
[1-({1-[(4-chloro-1-methyl-1H-pyrazol-3-yl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanamine
1-(3-chloro-4-fluorobenzenesulfonyl)-4-(1-methyl-1H-imidazol-2-yl)piperidine
3-benzyl-5-(butoxymethyl)-1H-1,2,4-triazole
N-[2-(furan-2-yl)ethyl]-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-{[(propan-2-yl)amino]methyl}piperidin-2-one
3-cyclobutyl-1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-phenylmethanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
N-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-(1H-pyrazol-3-yl)benzamide
2-{4-[benzyl(methyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}acetamide
2-(4-fluorophenyl)-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
N-[3-(4-chlorophenoxy)-2-hydroxypropyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
1-(4-methoxybenzoyl)-4-(thiophene-3-carbonyl)piperazine
1-{1-[3-(furan-2-yl)propanoyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
(3aS,6aS)-2-(2-cyclopentylacetyl)-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[5-(oxolan-2-yl)thiophen-2-yl]-1H-1,3-benzodiazole
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-(pyridin-2-ylmethyl)piperidine-4-carboxamide
1-[(3-{2-hydroxy-3-[methyl(propan-2-yl)amino]propoxy}-4-methoxyphenyl)methyl]piperidine-4-carbonitrile
4-(2-hydroxyethyl)-N-[4-(3-methoxyphenoxy)phenyl]piperazine-1-carboxamide
2-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-N,N-dimethylaniline
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-(pyrrolidin-1-ylmethyl)benzamide
(3S,4S)-4-(pyrrolidin-1-yl)-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-ol