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6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-1,3-benzodiazole
1-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-2-cyclobutyl-5-fluoro-1H-1,3-benzodiazole
3-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-fluoro-2-methylphenyl)urea
1-[4-(2-fluorophenyl)piperazin-1-yl]-3-(3-methylpiperidin-1-yl)propan-1-one
2-[(2E)-3-phenylprop-2-en-1-yl]-8-(thiophene-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-[1-(thiophen-2-yl)ethyl]acetamide
N-cyclopentyl-3-({[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl](methyl)carbamoyl}methyl)morpholine-4-carboxamide
1-methyl-N-(2-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1H-indazole-3-carboxamide
N-(1-{2-amino-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}piperidin-4-yl)pyridin-2-amine
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[2-oxo-2-(piperazin-1-yl)ethyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
6-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-2-methyl-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
N-[(4-chlorophenyl)(pyridin-3-yl)methyl]-2-methylpyrido[2,3-d]pyrimidin-4-amine
N-[(2,5-dichlorophenyl)methyl]-2-(1,4-dimethylpiperazin-2-yl)acetamide
N-[(2R,4R,6S)-2-cyclohexyl-6-[4-(1H-1,2,4-triazol-1-yl)phenyl]oxan-4-yl]acetamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)pyridazine-4-carboxamide
2-[4-(5-fluoropentyl)phenyl]-5-methyl-1,3,4-oxadiazole
6-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidine-1-carbonyl]-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
N-[(1-{[(1,5-dimethyl-1H-pyrazol-4-yl)carbamoyl]methyl}piperidin-3-yl)methyl]-4-fluorobenzamide
N-(9H-fluoren-9-yl)-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
4-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)pyridine
1-{3-[(3-fluorophenyl)amino]piperidin-1-yl}-2-(2-methoxyphenoxy)ethan-1-one
2-(3-hydroxypiperidin-1-yl)-1-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]ethan-1-one
N-[(3R,4S)-1-acetyl-4-(propan-2-yl)pyrrolidin-3-yl]-4-(4-fluorophenyl)butanamide
3-(2,4,5-trimethylbenzoyl)-3,9-diazaspiro[5.5]undecane
methyl 2-hydroxy-5-[6-oxo-3-(pyridin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl]benzoate
N-(cyclopent-3-en-1-yl)-1-(1-cyclopropanecarbonylpiperidin-4-yl)piperidine-3-carboxamide
N-(3-fluorophenyl)-3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
4-[2-(4-fluorophenoxy)ethyl]-1-(3-methylbenzoyl)-1,4-diazepan-5-one
2-(5-oxopyrrolidin-2-yl)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)acetamide
5-{[2-(carboxymethyl)piperidin-1-yl]methyl}-2-methoxybenzoic acid
1-(2-methanesulfonylethyl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1,4-diazepan-6-ol
3-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1-methyl-1H,2H,3H-imidazo[4,5-c]pyridin-2-one
(3aR,5R,6S,7aS)-2-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-octahydro-1H-isoindole-5,6-diol
methyl[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]{[5-(oxolan-2-yl)thiophen-2-yl]methyl}amine
1-{4-[2-(benzylsulfanyl)-4-hydroxypyrimidine-5-carbonyl]piperazin-1-yl}ethan-1-one
N-(1,3-benzothiazol-2-ylmethyl)-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3S,4R)-1-(1-benzofuran-5-carbonyl)-4-methyl-3-(2-methylpropyl)piperidin-4-ol
N-(3-{[(2,2-dimethyloxan-4-yl)(ethyl)carbamoyl]amino}-4-methylphenyl)-2-methoxyacetamide
N-(2-methoxyethyl)-3-[(3S,4R)-1-(pyridin-3-ylmethyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanamide
(3aR,5S,6S,7aS)-2-(1-tert-butyl-1H-pyrrole-3-carbonyl)-octahydro-1H-isoindole-5,6-diol
N-cyclopropyl-2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]pyridine-4-carboxamide
N-({1-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)acetamide
(1R,5S,6R)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-[(1-phenyl-1H-pyrazol-4-yl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
9-(3-methyl-1-benzothiophen-2-yl)-2H,3H,4H,6H,7H,8H,9H-[1,4]oxazino[2,3-g]quinoline-3,7-dione
2-benzyl-4-(5-fluoro-2-methylbenzenesulfonyl)morpholine
1-[(2-ethylpyrimidin-5-yl)methyl]-4-(piperidine-1-sulfonyl)-1,4-diazepane
3-(2,4-dimethoxybenzoyl)-1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidine
N-(oxolan-2-ylmethyl)-2-{4-[1-(pyridin-2-yl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}acetamide
3-[(3S,4R)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]-1-ethyl-6,7,8-trifluoro-1,4-dihydroquinolin-4-one
(1R,5S,6R)-3-cyclopropanecarbonyl-6-{[4-(2-phenylethyl)piperazin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane