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4-[(3S,4R)-4-hydroxyoxolan-3-yl]-N-[3-(1,3-thiazol-4-yl)phenyl]-1,4-diazepane-1-carboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(3-phenylpropyl)piperidine-4-carboxamide
{1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-4-yl}(thiophen-2-yl)methanol
5-{2-[2-(1H-imidazol-4-yl)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carbonyl}-1-methyl-1H-pyrrole-3-carbonitrile
(2R,3R,6R)-3-(4-methoxyphenyl)-5-[(4-methoxypyridin-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
5-benzyl-4-[3-(dimethylamino)propanoyl]-1-(3-methoxyphenyl)piperazin-2-one
N-[3-(methylsulfanyl)propyl]-3-[(piperidin-4-yl)sulfamoyl]benzamide
N-[(5,6-dimethylpyridin-3-yl)methyl]-1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-({[(3R,4R)-4-(hydroxymethyl)-1-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-carbonyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-[(3-fluorophenyl)methyl]-4-({[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}amino)pyrrolidin-2-one
2-methyl-5-{3-methyl-1-[(2-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl}-1,4-dihydropyridin-4-one
(3aR,5S,6S,7aS)-2-(5-phenoxyfuran-2-carbonyl)-octahydro-1H-isoindole-5,6-diol
5-ethyl-N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-(1-cyclohexyl-2,6,6-trimethyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(3-hydroxypropyl)acetamide
(3R,4R)-1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-4-cyclopropyl-3-methylpiperidin-4-ol
N,N-diethyl-1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-4-carboxamide
3-cyano-N-ethyl-N-[(2E)-3-phenylprop-2-en-1-yl]benzamide
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)[2-(3-methylpyridin-2-yl)ethyl]amine
3-(pyrimidin-5-yl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
5-(oxolan-2-yl)-3-(2-phenylethyl)-1H-1,2,4-triazole
(2S,4S,5R)-4-[(carboxymethyl)(methyl)carbamoyl]-5-(4-chlorophenyl)-1,2-dimethylpyrrolidine-2-carboxylic acid
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-oxopiperidine-3-carboxamide
8-(3-methylbutyl)-9-oxo-N-(propan-2-yl)-2,8-diazaspiro[5.5]undecane-2-carboxamide
N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1,3-thiazole-4-carboxamide
2-(4-{[methyl(oxan-4-yl)amino]methyl}phenyl)-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
2-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2,8-dimethylquinoline-4-carboxamide
3-[1-(6-aminopyridin-3-yl)-1H-1,3-benzodiazol-2-yl]propan-1-ol
N-[2-(1-hydroxycyclopentyl)ethyl]-5-(4-methoxyphenyl)furan-2-carboxamide
4-phenyl-1-[4-(1H-pyrazol-3-yl)benzoyl]-1,2,3,6-tetrahydropyridine
1-[(2-fluorophenyl)methyl]-N-methyl-N-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-amine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
5-methyl-2-[(oxolan-2-ylmethyl)sulfanyl]-4-{1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidin-3-yl}pyrimidine
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-6-methylphenol
1-oxo-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
[(3R,4R)-1-(3-chlorothiophene-2-carbonyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
1-cyclopentyl-N3-(2-hydroxy-2-phenylethyl)-N3-methyl-N5-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-(6-cyclopropylpyrimidin-4-yl)-4-[1-(methoxymethyl)cyclopropanecarbonyl]-1,4-diazepan-6-ol
4-[5-(1,4-dioxan-2-yl)-1-[(4-methylphenyl)methyl]-1H-1,2,4-triazol-3-yl]benzamide
2-(3-methoxypropyl)-8-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(2-oxopiperidin-1-yl)ethyl]acetamide
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)-5-[(dimethylamino)methyl]furan-2-carboxamide
3-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylpyridazine
N-ethyl-6-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N-methylpyrimidin-4-amine
1-[(5-chloro-2,4-dimethoxyphenyl)methyl]-4-(1-methyl-1H-imidazol-2-yl)piperidine
(5-{1-[(1-methylpiperidin-2-yl)methyl]-1H-imidazol-2-yl}furan-2-yl)methanol
5-(2-fluoro-4,5-dimethoxyphenyl)-1-[(3-fluorophenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazole
2-(4-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-1,3-benzothiazole
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine