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1-[(1S,5R)-6-(4-methoxy-2,3-dimethylbenzenesulfonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-{3-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]phenyl}imidazolidin-2-one
5-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,3-benzothiazol-2-amine
7-(5-chloro-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
4-{4-[1-(morpholin-4-yl)ethyl]phenyl}-6-(propan-2-yloxy)pyrimidin-2-amine
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-[(2S)-oxolan-2-ylmethyl]-1,2-oxazole-3-carboxamide
9-(quinoxalin-2-yl)-2H,3H,6H,7H,8H,9H-[1,4]dioxino[2,3-g]quinolin-7-one
2-benzyl-N-(3-ethylphenyl)-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxamide
1-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-3-(3-methoxy-4-methylphenyl)propan-1-one
2-cyclopropyl-N-{1-[(4-methylphenyl)methyl]cyclopropyl}-6-oxo-1,6-dihydropyrimidine-5-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[4-(3-methoxybenzoyl)piperazin-1-yl]ethan-1-one
6-fluoro-3-[2-(trifluoromethyl)morpholine-4-carbonyl]quinolin-4-ol
2-[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]-6-(5-methylthiophen-2-yl)pyridine-3-carboxylic acid
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-4-propylpyrimidine-5-carboxamide
N,N-dimethyl-4-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]piperidine-1-carboxamide
N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
1-[(3-fluorophenyl)methyl]-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperazine
N-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]naphthalene-1-carboxamide
3-hydroxy-1-(3-phenylpropyl)-3-[(4-propylpiperazin-1-yl)methyl]piperidin-2-one
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(4-hydroxybutyl)pyrrolidine-3-carboxylic acid
2-{5-[(2,4,6-trifluorophenyl)methyl]-1,2,4-oxadiazol-3-yl}pyrazine
N-[2-(morpholin-4-yl)propyl]-1-(pyridin-2-ylmethyl)piperidin-4-amine
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-N-methyl-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-(3,5-difluorophenyl)-N-[(4,5-dimethylfuran-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
4-ethyl-1-[(4-methylbenzenesulfonyl)methyl]-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[3-(2-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-3-(1H-pyrazol-1-yl)benzamide
2-(carbamoylamino)-N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methylacetamide
4,5-dimethyl-2-(2-{4-[1-(propan-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-1-yl}ethyl)-1H-1,3-benzodiazole
4-(1H-imidazol-1-yl)-1-[2-(oxolan-2-ylmethoxy)acetyl]piperidine-4-carboxylic acid
N'-(5-methyl-1,2-oxazol-3-yl)-N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)ethanediamide
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
N-[(1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-3-yl)methyl]methanesulfonamide
3-(1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3-carbonyl)pyridine
6-(2,5-dimethylfuran-3-yl)-7-methyl-2-(4-methylpiperazine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
methyl (2S,4S)-1-methyl-4-(5-phenyl-1H-pyrrole-2-amido)pyrrolidine-2-carboxylate
3-{[methyl(prop-2-en-1-yl)amino]methyl}-N-(1-methyl-1H-pyrazol-4-yl)benzamide
2-[(dimethylcarbamoyl)amino]-N-[3-(pyridin-4-yl)propyl]acetamide
1-(3-methylpyridin-4-yl)-4-(1-phenylcyclopropanecarbonyl)-1,4-diazepane
2-[3-hydroxy-3-(hydroxymethyl)piperidine-1-carbonyl]-5,7-dimethylquinolin-8-ol
1-[1-(1,4-dithiepan-6-yl)piperidin-3-yl]-4-(4-methoxyphenyl)piperazine
N-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(4-methylphenyl)ethan-1-one
7-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2,3,4-tetrahydroquinoxalin-2-one
3-[(3R,4S)-1-(isoquinoline-5-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
1-[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-cyclopropylethan-1-one
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-(morpholin-3-yl)acetamide
1-(carbamoylmethyl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}piperidine-3-carboxamide
N-methyl-5-{[4-(naphthalen-2-yl)-1H-1,2,3-triazol-1-yl]methyl}furan-2-carboxamide
1-(1-methyl-5-{[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1H-pyrrol-3-yl)ethan-1-one
N-(2-methyl-1-benzofuran-7-yl)-1H-indazole-3-carboxamide