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6-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]pyridine-3-carboxylic acid
N-{2-[5-methyl-4-(propanamidomethyl)-1,3-oxazol-2-yl]phenyl}-3-phenoxypropanamide
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-5-[(2-methoxyethyl)sulfanyl]-1,3,4-thiadiazol-2-amine
2-(benzyloxy)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}acetamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]butane-1-sulfonamide
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-N-[1-(1H-indol-5-yl)ethyl]propanamide
(4aS,8aR)-6-(5-methyl-1,2-oxazole-3-carbonyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
4-{6-[4-(thiophen-2-ylmethyl)piperazin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}morpholine
N-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]benzamide
2-(2-aminopyrimidin-5-yl)-N,8-dimethyl-N-[1-(pyridin-2-yl)propan-2-yl]quinoline-4-carboxamide
5-{2-[4-(2-fluorophenoxy)piperidin-1-yl]-2-oxoethyl}-1,3-dimethylimidazolidine-2,4-dione
2-({5-[1-(1H-pyrazol-1-yl)ethyl]-4-(pyridin-3-yl)-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
N-(1-{2-[3-methyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1H-indol-3-yl}propan-2-yl)acetamide
1-(3-fluorophenyl)-4-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidin-3-amine
3-fluoro-5-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
2-(5-fluoro-2-methoxyphenyl)quinoline
thiophen-2-yl({1-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]piperidin-4-yl})methanol
1-{2-[4-(benzyloxy)piperidin-1-yl]-2-oxoethyl}piperidine-4-carboxamide
2-[1-(furan-3-ylmethyl)-1H-1,2,3-triazol-4-yl]-1-(2-methylpropyl)-1H-1,3-benzodiazole
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-4-(1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-amine
3-{2-[4-(4-acetylphenyl)piperazin-1-yl]-2-oxoethyl}-5,5-dimethyl-1,3-oxazolidine-2,4-dione
3-({2-[2-methyl-1-(morpholin-4-yl)propan-2-yl]-1H-imidazol-1-yl}methyl)quinoline
3-(1H-pyrazol-1-ylmethyl)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]benzamide
N-(propan-2-yl)-1-[(1s,4s)-4-(5-methyl-3-phenyl-1,2-oxazole-4-amido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-[(3-methoxyphenyl)amino]-N-[2-(pyridin-3-yl)ethyl]butanamide
2-[3-cyclopropyl-1-(4-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]-3-fluoropyridine
1,9-dimethyl-4-[2-(2-methyl-1H-1,3-benzodiazol-1-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-cyclobutyl-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
2-amino-7-(2,3-dimethoxybenzoyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-[1-(2,3-dihydroxypropyl)-4-phenyl-1H-imidazol-5-yl]-1-methyl-1,2-dihydroquinolin-2-one
2-phenyl-5-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}-2,3-dihydro-1H-pyrazol-3-one
(2R)-2-amino-3-(1H-indol-3-yl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)propanamide
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
4-chloro-2-{[methyl({[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}phenol
3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]benzamide
3-{1-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]piperidin-3-yl}-N-(4-fluoro-2-methylphenyl)propanamide
2-butoxy-1-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}ethan-1-one
(4aS,7aR)-1-{[2-(ethylamino)pyrimidin-5-yl]methyl}-4-(1H-imidazol-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-methyl-N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]imidazo[1,2-a]pyridine-6-carboxamide
5-{5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}-2-methyl-1H-pyrrole-3-carbonitrile
N,N-dimethyl-2-{1H,3H,4H,5H-thiopyrano[4,3-b]indol-8-ylformamido}propanamide
N-[4-(1H-pyrazol-1-yl)phenyl]-1-(thiophen-3-ylmethyl)piperidine-4-carboxamide
2-ethyl-1-[9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butan-1-one
N-[2-(4-chlorophenyl)-2-(pyrrolidin-1-yl)ethyl]-2-(dimethylamino)-4-methylpyrimidine-5-carboxamide
2-{[5-(3-acetylphenoxymethyl)-1H-pyrazol-3-yl]formamido}acetamide
(1R,2R,6S,7S)-4-[5-(methanesulfonylmethyl)pyridin-2-yl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-3,5,7-trimethyl-1H-indole-2-carboxamide
4-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]phenol
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide