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N-{[7-chloro-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-1,3-thiazole-5-carboxamide
[(3S,4S)-4-(hydroxymethyl)-1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)pyrrolidin-3-yl]methanol
(1R,5R)-6-(5-chloro-2-methoxybenzoyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
4-ethyl-4-({[2-methyl-1-(pyrrolidin-1-yl)propan-2-yl]amino}methyl)hexanenitrile
3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-4-ylmethyl)propanamide
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylpyridine-4-carboxamide
(1R,2S,6R,7S)-4-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-4-azatricyclo[5.2.2.02,6]undecane
6-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1-(4-methylphenyl)urea
1-(3-{[(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amino]methyl}phenyl)ethan-1-one
1-(oxolane-3-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
1-ethyl-3-methyl-4-[2-(pyridin-3-yloxy)acetyl]piperazin-2-one
2-(methylsulfanyl)-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]pyridine
6-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
(1S,5R)-3-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-{[(oxan-4-yl)amino]methyl}piperidin-2-one
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]spiro[2.4]heptane-1-carboxamide
(2S)-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-2,3-dihydro-1H-indole-2-carboxamide
1-(2-{[2-(5-propylfuran-2-yl)-1H-imidazol-1-yl]methyl}morpholin-4-yl)ethan-1-one
2-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine-4-carboxamide
2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]-N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)acetamide
(3S,9aR)-2-methyl-8-(3-methylbutyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(cyclopent-2-en-1-yl)-N-(furan-2-ylmethyl)-N-(prop-2-en-1-yl)acetamide
(1S,4S)-2-(2,3-dihydro-1H-inden-5-yl)-5-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-2,5-diazabicyclo[2.2.1]heptan-3-one
2-methyl-2-{5-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-4-phenyl-1H-imidazol-1-yl}propane-1,3-diol
N-(3-hydroxypropyl)-1-(4-methoxyphenyl)-2,2-dimethylcyclopropane-1-carboxamide
N-{2-[1-(5-fluoro-2-methylphenyl)-1H-imidazol-4-yl]ethyl}acetamide
1-{2-[({4-[2-hydroxy-3-(thiomorpholin-4-yl)propoxy]-3-methoxyphenyl}methyl)amino]ethyl}imidazolidin-2-one
4-[4-(furan-3-carbonyl)-1,4-diazepane-1-carbonyl]-2,3,6-trimethylquinoline
methyl 1-{2,6-dimethylimidazo[1,2-a]pyridine-3-carbonyl}pyrrolidine-2-carboxylate
(3S,4R)-1-{2-[(3-methoxyphenyl)sulfanyl]acetyl}-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
4-(pyrimidin-2-yl)-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperazine-2-carboxylic acid
N,N-diethyl-1-[5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carbonyl]pyrrolidin-3-amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
(2S,4S)-4-(4-cyanobenzamido)-N,1-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidine-2-carboxamide
2-[1-(3-phenyl-1H-1,2,4-triazol-5-yl)propyl]-2,3-dihydro-1H-isoindol-1-one
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-3-{[(3R)-pyrrolidin-3-yl]sulfamoyl}benzamide
N-{4-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-2-(5-oxopyrrolidin-2-yl)acetamide
7-[(2-fluorophenyl)methyl]-2-(thiophene-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-{[methyl({[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}pyridin-2-amine
(1R,5R)-3-benzoyl-6-[3-(benzyloxy)propyl]-3,6-diazabicyclo[3.2.2]nonane
4-(1,5-dimethyl-1H-pyrazole-4-carbonyl)-1-methyl-1,4,9-triazaspiro[5.5]undecane
1-methyl-3-(1-{2-[methyl(propan-2-yl)amino]acetyl}piperidin-3-yl)-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-6-fluoro-2-(1-propyl-1H-pyrazol-4-yl)quinoline
4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-2-[(3-methoxyphenyl)methyl]morpholine
2-(4-{1-[(3-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-1-yl)-N-(propan-2-yl)acetamide
5-{[4-(4-chlorophenyl)butanamido]methyl}-N,N-dimethylfuran-2-carboxamide
2-(oxolan-2-ylmethyl)-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)(methyl){[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}amine