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N-methyl-4-(2-methyl-1H-imidazol-1-yl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]butanamide
methyl(3-{4-[4-(trifluoromethoxy)phenyl]-1H-1,2,3-triazol-1-yl}propyl)amine
2-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-methoxypyrazine
1-benzyl-3-(2-methoxyphenyl)-6-(pyridin-4-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
3-[(3,3-dimethylcyclohexyl)amino]-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-5-[(propan-2-yl)sulfamoyl]benzamide
N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
1-(4-{5-methoxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}phenyl)pyrrolidin-2-one
N-(2-hydroxypropyl)-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(2-fluorophenyl)propan-1-one
4-(3-chloro-4-fluorobenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl){[1-(morpholin-4-yl)cyclohexyl]methyl}amine
(1R,9S)-5-amino-3-(3-cyanophenyl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
3-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-4,5,6,7-tetrahydro-1H-indazole
methyl 7-(2-chlorobenzamido)-1,2,3,4-tetrahydroisoquinoline-2-carboxylate
2-(4-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}morpholin-2-yl)ethan-1-ol
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-3-(dimethylamino)piperidine-1-carboxamide
N-{1-[1-(3-cyano-2-methoxypyridin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
(3-{2-azabicyclo[2.2.1]hept-5-en-2-yl}propyl)({[7-fluoro-2-(morpholin-4-yl)quinolin-3-yl]methyl})amine
2-[3-(3-fluorophenoxymethyl)piperidin-1-yl]-4-(1-methyl-1H-pyrazol-4-yl)pyrimidine
2-(2-hydroxyethyl)-9-(3,4,5-trifluorobenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{[2-(2-hydroxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]methyl}benzonitrile
7-(propan-2-yl)-2-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
3-(methylsulfanyl)-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
9-[4-(pyridin-4-yl)piperidin-1-yl]-3-azaspiro[5.5]undecane
2-(1,2-oxazol-5-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(4-methyl-1,4-diazepan-1-yl)ethan-1-one
5-[9-hydroxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(4-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
(4aR,7aS)-4-(2-hydroxypyridine-3-carbonyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-{[methyl(propyl)amino]methyl}piperidin-2-one
3-methyl-1-[3-(pyridin-3-yl)azetidin-1-yl]-2-[(quinazolin-4-yl)amino]butan-1-one
N-[(5-carbamoyl-1,2,4-oxadiazol-3-yl)methyl]-2-ethylpyrimidine-5-carboxamide
3-[(3-methylbutyl)amino]-N-[(3S)-2-oxoazepan-3-yl]-5-[(propan-2-yl)sulfamoyl]benzamide
3-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-1-[2-(furan-2-ylmethyl)-3-hydroxypropyl]urea
2-oxo-6-(propan-2-yl)-N-{2-[(trifluoromethyl)sulfanyl]ethyl}-1,2-dihydropyridine-3-carboxamide
1-({3-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methyl)-1H-1,3-benzodiazole
4-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
2-[1-(2-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(2-hydroxyethyl)-N-methylacetamide
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-[(1-methyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-{2-[3-(4-methylpiperazin-1-yl)-3-oxopropyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-2,3-dihydro-1H-imidazol-2-one
2-(thiophen-3-ylmethyl)-4-(4-{[4-(trifluoromethyl)phenyl]methyl}piperazin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
methyl 2-({[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)benzoate
4-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)morpholine
2-[1-({1-[(1-methyl-1H-indol-3-yl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
4-[(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]-1,5-dimethyl-1H-pyrrole-2-carbonitrile
3-chloro-6-[3-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridazine
(cyclohex-3-en-1-ylmethyl)({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
(3S,4R)-4-methyl-1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}piperidine-3,4-diol
6-ethyl-2-(morpholin-4-yl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidin-4-amine
2-chloro-4-{[(2-hydroxyethyl)({[4-(methylsulfanyl)phenyl]methyl})amino]methyl}-6-methoxyphenol