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4-[2-(dimethylamino)benzoyl]-1-(4-methylphenyl)piperazin-2-one
N-(3,4-dimethylphenyl)-1-(4-methylbenzoyl)piperidin-3-amine
1-cyclopentyl-4-[({5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}amino)methyl]pyrrolidin-2-one
N-(1-benzothiophen-5-ylmethyl)-2-(2-oxopyrrolidin-1-yl)propanamide
2-[1-(cyclohexylmethyl)-4-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}piperazin-2-yl]ethan-1-ol
N-methyl-N-(2-{[4-(pyridin-4-yl)pyrimidin-2-yl]amino}ethyl)methanesulfonamide
2-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
2,5-dimethyl-3-{4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}pyrazine
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
N-(4-{[1-(3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}phenyl)acetamide
1-[benzyl(methyl)amino]-3-[2-methoxy-5-({[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
N-[(5-methylfuran-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
3-[4-(1-methyl-1H-indole-6-carbonyl)piperazin-1-yl]-1λ6-thiolane-1,1-dione
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-propyl-N-(pyridin-4-ylmethyl)acetamide
N-methyl-2-(phenoxymethyl)-N-[1-(thiophen-2-yl)ethyl]-1,3-oxazole-4-carboxamide
methyl 2-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}butanoate
4-(4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-1-yl)-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
1-methyl-2-oxo-8-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-cyclohexyl-N-[2-(1H-indol-3-yl)ethyl]oxolane-3-carboxamide
2-(4-chloro-2-methylphenoxy)-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}propanamide
3,5-dimethyl-1-{1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]pyrrolidin-3-yl}-1H-pyrazole
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}pyrazine-2-carboxamide
6-{3-[3-(4-methoxy-2-methylbenzoyl)piperidin-1-yl]-3-oxopropyl}-2,3,4,5-tetrahydropyridazin-3-one
(3S,4R)-3-acetamido-N-(5-fluoro-2-methylphenyl)-4-propylpyrrolidine-1-carboxamide
1-[(3,4-dimethylphenyl)methyl]-4-(6-methoxypyrimidin-4-yl)piperazin-2-one
4-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
7-(ethanesulfonyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[1-(cyclopentylmethyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
2-oxo-N-[2-(3-phenylpiperidin-1-yl)ethyl]-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
(2S,4R)-1-[(2-chlorophenyl)methyl]-4-{[(4-fluorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
1-(4-fluorobenzoyl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
2-({6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]quinazolin-4-yl}amino)ethan-1-ol
1-[(3-fluorophenyl)methyl]-4-{[5-(oxan-2-yl)thiophen-2-yl]methyl}piperazine
2-methoxy-N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]pyridine-4-carboxamide
N-[3-(2-methoxyphenyl)propyl]thian-4-amine
ethyl 2-{1-[(4-{[(5-methylfuran-2-yl)methyl]amino}quinazolin-2-yl)methyl]piperidin-2-yl}acetate
3-[({1-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]piperidin-4-yl}amino)methyl]-1λ6-thiolane-1,1-dione
N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
5-[1-(2-hydroxyethyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
3-fluoro-4-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)pyridine
(1R,4S)-1,7,7-trimethyl-4-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]-2-oxabicyclo[2.2.1]heptan-3-one
1-[2-(1H-imidazol-4-yl)ethyl]-4-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-1,2,3-triazole
2-{4-[4-(ethylamino)pyrimidin-2-yl]phenyl}acetic acid
3-(1,4-dioxan-2-ylmethyl)-1-(3-methylbutyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
N-(3-ethoxypropyl)-5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carboxamide
(1-{5-cyclopropyl-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperidin-4-yl)methanol
N-({1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]pyrrolidin-3-yl}methyl)-5-methylpyrazine-2-carboxamide
ethyl 1-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-4-(2-phenylethyl)piperidine-4-carboxylate
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[3-(4-fluorophenyl)-4-methyl-1H-pyrazol-1-yl]acetamide