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1-{[2-amino-6-(pyrrolidin-1-yl)pyrimidin-4-yl]amino}-3-(azepan-1-yl)propan-2-ol
1-[2-chloro-5-(pyrrolidine-1-carbonyl)phenyl]-3-[3-(1H-imidazol-1-yl)propyl]urea
4-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-3-yl]-5-methyl-2-[(oxolan-2-ylmethyl)sulfanyl]pyrimidine
N,6-dimethyl-2-oxo-4-(pyridin-3-yl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-(carbamoylmethyl)-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methylpiperidine-3-carboxamide
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]furan-2-carboxamide
1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-4-phenoxybutan-1-one
6,7-dimethoxy-2-[1-(1-propylpiperidin-4-yl)piperidin-3-yl]-1,2,3,4-tetrahydroisoquinoline
1-(5-{2-amino-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}-2-methylphenyl)imidazolidin-2-one
[3-(cyclopropylmethyl)-1-(2-methanesulfonylethyl)piperidin-3-yl]methanol
(1R,5S,6R)-N,N-diethyl-6-{[(furan-3-ylmethyl)(methyl)amino]methyl}-3-azabicyclo[3.1.0]hexane-3-carboxamide
({5-[1-(5-chloropyridine-2-carbonyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-4-(oxolane-2-carbonyl)-1,4-diazepane
2-{2-benzyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-N-methylpyridine-4-carboxamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-[(3-fluoropyridin-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
2,5-dimethyl-3-[4-(pyridin-4-yl)piperidin-1-yl]pyrazine
5-(3-acetylphenoxymethyl)-N-cycloheptyl-N-methyl-1H-pyrazole-3-carboxamide
N-methyl-2-(4-phenyl-5-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-imidazol-1-yl)butanamide
4-[hydroxy(thiophen-2-yl)methyl]-N-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]piperidine-1-carboxamide
N-[2-(4-methoxyphenyl)ethyl]-2,6-dimethyl-N-(pyridin-2-ylmethyl)pyridine-4-carboxamide
3-[1-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)piperidin-3-yl]-N-(4-fluoro-2-methylphenyl)propanamide
propan-2-yl N-{[1-(1H-1,3-benzodiazole-5-carbonyl)-4-hydroxyazepan-4-yl]methyl}carbamate
2-{[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]methyl}-6-methoxyphenol
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-3-phenyl-1H-pyrazole-4-carboxamide
N-phenyl-5-[(2S)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl]pyrimidin-2-amine
1-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]azetidin-3-ol
1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-2-(1,3-thiazol-2-yl)piperidine
methyl 9-(2,3-dihydro-1H-inden-2-yloxy)-7-oxo-3-(thiolan-3-yl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
[(2E)-2-methylbut-2-en-1-yl][(1-methylpiperidin-4-yl)methyl](2-phenylethyl)amine
2-{1-[(2-methylphenyl)methyl]-4-(quinolin-6-ylmethyl)piperazin-2-yl}ethan-1-ol
1-(morpholin-4-yl)-3-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]propan-1-one
1-(methoxymethyl)-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)cyclobutane-1-carboxamide
(3aR,5R,6S,7aS)-2-(4-phenylbenzenesulfonyl)-octahydro-1H-isoindole-5,6-diol
2-[cyclopentyl(methyl)amino]-1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)ethan-1-one
2,4-difluoro-N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)benzene-1-sulfonamide
1-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]-4-(4-methoxyphenyl)butan-1-one
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
1-(1-cyclopropanecarbonylpiperidine-4-carbonyl)-4-methoxy-4-phenylpiperidine
6-methyl-4-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}-1,2-dihydroquinolin-2-one
3-[2-(3-fluoro-2,4-dimethylphenyl)-1H-imidazol-1-yl]benzamide
4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(1-propyl-1H-indazol-3-yl)-2-[3-(thiophen-3-yl)-1H-pyrazol-1-yl]acetamide
5-methyl-1-{2-oxo-2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1R,5R)-N,N-dimethyl-6-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
11-{methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}-4-(3-phenylpropyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
6-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carboxamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}methanesulfonamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
N-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-N-(pyridin-4-ylmethyl)cyclopropanamine