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N-{2-[(4-chlorophenyl)methoxy]ethyl}-3-methyl-4-oxo-3,4-dihydroquinazoline-7-carboxamide
(4aS,8aS)-2-cyclopentanecarbonyl-7-(5-ethyl-1H-pyrrole-2-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
2-[(3,4-dimethoxyphenyl)methyl]-6-(3-propoxypiperidine-1-carbonyl)-1,3-benzoxazole
8-(5-chloro-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
6,7-dimethyl-4-[2-(morpholin-4-ylmethyl)phenyl]-1,3-benzothiazol-2-amine
3-(5-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}thiophen-2-yl)-1H-pyrazole
4-(5-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)pyridine
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
N-(oxolan-2-ylmethyl)-1-phenyl-N-(thiophen-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
7-(5-chloropyridin-2-yl)-4-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3S,4S)-1-(1-aminocyclopropanecarbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
diethyl[(5-methyl-4-{8-methyl-2,8-diazaspiro[4.5]decane-2-carbonyl}furan-2-yl)methyl]amine
5-fluoro-N-[3-(1H-1,2,3-triazol-1-yl)propyl]quinazolin-4-amine
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-(2-acetamidoethyl)-1-[(4-hydroxyphenyl)methyl]piperidine-3,5-dicarboxamide
2-ethyl-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]pyrimidine-5-carboxamide
(3aS,6aS)-2-methanesulfonyl-5-(1-methyl-1H-pyrrole-2-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-4-phenylpiperidin-4-yl]ethan-1-one
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-1-methyl-1H-indole-6-carboxamide
1-benzoyl-4-(2-fluoro-5-methylphenoxy)piperidine-4-carboxylic acid
1-(2-{[bis(prop-2-en-1-yl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
1-[(2-chlorophenyl)methyl]-N-(1,2-oxazol-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
6-chloro-3-{[(2,2-diphenylethyl)amino]methyl}-N,N-dimethylimidazo[1,2-a]pyridine-2-carboxamide
2-[2-({1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}methyl)phenoxy]ethan-1-ol
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]acetamide
(3aR,6aR)-2-cyclopropanecarbonyl-5-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-(2-amino-1,3-thiazol-4-yl)-N-methyl-N-(quinolin-3-ylmethyl)propanamide
2-(ethylamino)-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
5-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}-2-methoxyphenol
2-(3-{[3-(3-methylphenoxy)azetidin-1-yl]methyl}phenoxy)acetamide
8-benzyl-3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-cyclohexyl-5-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazol-5-yl]-3-ethyl-1H-1,2,4-triazole
N-({1-[(3-methoxyphenyl)methyl]pyrrolidin-3-yl}methyl)-1-methyl-1H-imidazole-5-carboxamide
2-ethoxy-5-[2-(morpholin-4-yl)pyrimidin-4-yl]benzoic acid
2-(dimethyl-1,3-thiazol-5-yl)-N-[3-(4-hydroxyphenyl)propyl]acetamide
N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}acetamide
4-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-(1-methyl-1H-pyrazol-5-yl)-4-({2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)benzamide
[1-(2,6-diaminopyrimidin-4-yl)-4-[(3-methoxyphenyl)methyl]piperidin-4-yl]methanol
5-{2-[(2-phenoxyethyl)amino]ethyl}-1-{[2-(trifluoromethoxy)phenyl]methyl}pyrrolidin-2-one
1-(3-propyl-1H-pyrazole-5-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperazine
2-cyclopropyl-5-[4-(3,4-dichlorophenyl)piperazine-1-carbonyl]pyrimidine
2-[(3,5-difluorophenyl)methyl]-8-(4-methylbenzoyl)-2,8-diazaspiro[4.5]decan-3-one
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-amine
1-{3-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
[(3R,4R)-1-(2-ethylbenzoyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
(4aS,8aR)-2-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]-decahydroisoquinoline
2-[4-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-5-methylphenol
1-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(pyrazin-2-yl)propan-1-one
(7R,9aR)-N-(3-fluorophenyl)-7-(hydroxymethyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide