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[(3R,4R)-4-(morpholin-4-ylmethyl)-1-(1,3-oxazole-4-carbonyl)pyrrolidin-3-yl]methanol
3-(5-{[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1-(propan-2-yl)-1H-pyrazole
1-[2-(4-chlorophenyl)ethyl]-N-[(4-methylphenyl)methyl]-6-oxopiperidine-3-carboxamide
3-{[benzyl(methyl)amino]methyl}-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
7-methyl-3-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]-3,7,11-triazaspiro[5.6]dodecan-12-one
2-fluoro-6-({[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amino}methyl)phenol
4-(4-chlorophenyl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]butanamide
2-(1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)propan-2-ol
N-[3-(4-{[3-(1H-1,2,3-benzotriazol-1-yl)propyl]amino}piperidin-1-yl)phenyl]-4-phenylbutanamide
{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
5-{[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}-2-(3-methylphenyl)pyrimidine
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[(1-methyl-1H-imidazol-5-yl)methyl]piperidine-4-carboxamide
N-[2-(4H-1,2,4-triazol-4-yl)ethyl]-5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-amine
3,5-dimethyl-4-(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}pyrrolidin-2-yl)-1,2-oxazole
N-{2-[1-(8-hydroxy-5,7-dimethylquinoline-2-carbonyl)piperidin-2-yl]ethyl}acetamide
N-({1-[(3-fluoropyridin-4-yl)methyl]pyrrolidin-3-yl}methyl)-2-hydroxypyridine-3-carboxamide
4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-N,6-dimethylpyrimidin-2-amine
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(4-fluorophenyl)piperidin-4-ol
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-(naphthalen-1-yl)ethyl]acetamide
6-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)pyridine-3-carboxylic acid
1-(4-{[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
3-(3,4-difluorophenyl)-1-(6-hydroxy-1,4-oxazepan-4-yl)propan-1-one
2-{1-[2-(ethanesulfonyl)ethyl]-1H-imidazol-2-yl}pyridine
1-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
N-cyclopentyl-1-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-1H-pyrazole-5-carboxamide
(1R,3S)-3-[4-(pyridin-4-yl)piperazine-1-carbonyl]cyclopentan-1-amine
{2-[4-(4-methylpiperazin-1-yl)quinazolin-6-yl]phenyl}methanol
2-(pentafluoroethyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
8-methoxy-2-{[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}quinoline
(1S,5R)-6-(pyrazine-2-carbonyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-(1H-pyrrole-2-carbonyl)piperazine
5-butyl-1'-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(4-tert-butylphenoxymethyl)-4-hydroxy-N-[1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]pyrimidine-5-carboxamide
3,5-dimethyl-4-oxo-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
1-(1-methyl-1H-pyrrole-2-carbonyl)-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
3-[2-(2,6-difluorophenyl)ethyl]-1-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}piperidine
1,3-dimethyl-6-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
[(3R,4R)-1-[(5-methylfuran-2-yl)methyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
1-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-2-(oxolan-3-yl)-1H-imidazole
1-methyl-N-[2-(phenylsulfanyl)ethyl]-N-(prop-2-en-1-yl)-1H-pyrrole-2-carboxamide
3-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-1-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
4-[4-(dimethylamino)phenyl]-3-phenyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(3R)-1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-3,4,4-trimethylpyrrolidin-3-ol
3-[5-(2-ethoxyethyl)-1,3,4-thiadiazol-2-yl]-1-[1-(1H-imidazol-1-yl)butan-2-yl]urea
3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]-N-(2,2,2-trifluoroethyl)propanamide
5-acetyl-2,4-dimethyl-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-pyrrole-3-carboxamide
5-chloro-2-(2-ethylmorpholine-4-carbonyl)-3-phenyl-1H-indole
(1R,5R)-3-(5-ethylthiophene-2-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane