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[(4aS,8aR)-6-{[5-(1,2-oxazol-3-yl)thiophen-2-yl]sulfonyl}-decahydro-1,6-naphthyridin-4a-yl]methanol
2-(4-fluorophenyl)-N-methyl-N-[1-(pyridin-2-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
2-[3-({4-[(2,2-dimethylpyrrolidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}methyl)piperidine-1-carbonyl]pyridin-4-amine
N-[(2-fluorophenyl)methyl]-2-({2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}amino)acetamide
1-(3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}pyrrolidin-1-yl)-3-methylbutan-1-one
1'-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
6-{[1-(cyclohexylmethyl)piperidin-3-yl]amino}-N,N-dimethylpyridine-3-carboxamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-5-propyl-1,3,4-oxadiazol-2-amine
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-4-(1H-1,2,4-triazol-1-yl)butanamide
N-[2-methyl-1-(7-{[3-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)propyl]methanesulfonamide
3-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-methylpropanamide
1-[2-(2-chlorophenyl)ethyl]-N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(methoxymethyl)-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
dimethyl({5-[4-(3-phenylpropyl)piperidine-1-carbonyl]-1,3,4-oxadiazol-2-yl}methyl)amine
4-acetyl-N-[4-(3-methylpiperidine-1-carbonyl)phenyl]-1,4-diazepane-1-carboxamide
N-benzyl-N-methyl-3-[1-(6-oxopiperazine-2-carbonyl)piperidin-4-yl]propanamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
6-[3-(2-methylphenoxymethyl)piperidine-1-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
4-methyl-2-({4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)phenol
N-[(1-benzylpyrrolidin-3-yl)methyl]-4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N'-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]pentanediamide
N-butyl-2-({6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}(methyl)amino)acetamide
N-({7-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
{[5-(furan-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}(methyl){[3-(methylsulfanyl)phenyl]methyl}amine
2-[4-(2-aminopyrimidin-4-yl)-1H-pyrazol-1-yl]-N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
6-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-5-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-tert-butyl-N-{[3-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidine-3-carboxamide
9-(2,6-dimethylpyridin-4-yl)-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}ethan-1-one
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
2-[(1-benzyl-4-phenylpiperidin-4-yl)formamido]acetic acid
1-{3-[2-(pyridin-3-yl)-1H-imidazol-1-yl]phenyl}ethan-1-ol
1-[2-(4-methoxyphenyl)ethyl]-8-[(1-methyl-1H-indol-3-yl)methyl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(2,3-difluoro-4-methoxyphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]acetamide
4-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
2-[(1S,5R)-6-{[4-(3-hydroxyprop-1-yn-1-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
N,N-dimethyl-5-[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]-1,2,4-thiadiazol-3-amine
1-cyclohexyl-4-(3-methyl-1,2,4-oxadiazol-5-yl)piperidine
1-[(2-methylphenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(3aR,7aS)-2-(3-propyl-1H-pyrazole-5-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
N,N,5-trimethyl-2-[3-(1H-pyrazol-3-yl)phenyl]pyrimidin-4-amine
1-{4-[2-(cyclopentylmethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}propan-1-one
1-cyclopentyl-4-[2-(morpholin-4-yl)ethyl]-1,4-diazepane-6-carboxylic acid
[1-(1,4-dithiepan-6-yl)-3-(3-phenylpropyl)piperidin-3-yl]methanol
1-(2,3-dihydro-1H-inden-5-yl)-5-[(2-methoxyethoxy)methyl]-1H-1,2,4-triazole
N-(1-methoxypropan-2-yl)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-(morpholin-4-yl)-1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]propan-1-one
1-{[(3R,4R)-1-(4-chlorobenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
7-[(2-phenyl-1,3-oxazol-4-yl)methyl]-2-oxa-7-azaspiro[4.5]decan-8-one
methyl 5-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-5-oxopentanoate