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N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
5-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]pyridin-3-amine
[(1-{[1-(thian-4-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]urea
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-methyl-6-(propan-2-yl)pyrimidin-4-amine
N-[1-(4-ethoxy-3-fluorophenyl)ethyl]-5-methanesulfonyl-2-methylpyrimidin-4-amine
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[2-methyl-2-(morpholin-4-yl)propyl]-1H-pyrazole-3-carboxamide
3-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-ylmethyl]-4-chloro-1-methyl-1H-indazole
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-methoxy-2-methylpropan-1-one
N2-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N4,N4,5-trimethylpyrimidine-2,4-diamine
4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-[(3-methoxyphenyl)methyl]piperazin-2-one
2-(1-{[5-(2-chlorophenyl)furan-2-yl]methyl}piperidin-4-yl)-N-methylacetamide
[(3S,5R)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(1H-1,2,3-triazole-5-carbonyl)piperidin-3-yl]methanol
2-(2,5-dioxoimidazolidin-1-yl)-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)acetamide
1-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(thiophen-2-yl)ethan-1-one
N-{1-[1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carbonyl]piperidin-4-yl}acetamide
8-[1-methyl-3-(trifluoromethyl)-1H-thieno[2,3-c]pyrazole-5-carbonyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
1-{[5-(4-methoxyphenyl)furan-2-yl]methyl}-4-(pyridin-3-yl)piperazine
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-N-methyl-4-{[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]amino}pyrrolidine-2-carboxamide
N-[3-(benzylsulfanyl)propyl]-1-ethylpiperidine-3-carboxamide
3-[6-oxo-2-(pyrrolidin-1-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-8-yl]-1,2-dihydroquinolin-2-one
1-{4-[3-(1H-pyrazol-3-yl)phenyl]phenyl}propan-1-ol
N-[5-({4-[(4-methylphenyl)methyl]-5-oxo-1,4-diazepan-1-yl}methyl)thiophen-2-yl]acetamide
1-[2-(5-chloro-2-methoxyphenyl)pyrimidin-4-yl]piperidin-3-ol
N-{[1-(1,3-thiazol-2-ylmethyl)piperidin-3-yl]methyl}naphthalene-1-carboxamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-(trimethyl-1H-pyrazol-1-yl)acetamide
N-cyclopropyl-1-[(3-methoxyphenyl)methyl]-5-(1,3-thiazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-methyl-5-{1-[4-(trifluoromethoxy)phenyl]-1H-1,2,4-triazol-5-yl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-propyl-1'-(5-propyl-1,2-oxazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(1R,5R)-N,N-dimethyl-6-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
(1R,5R)-6-[(4-methoxypyridin-2-yl)methyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
methyl 4-[5-({ethyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-1,2,4-oxadiazol-3-yl]benzoate
2-(2-methoxyethyl)-9-(4-phenylbutanoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(3-ethylphenyl)-4-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]-4-oxobutanamide
N-ethyl-N-(2-hydroxyethyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
4-fluoro-3-methyl-N-{[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}benzene-1-sulfonamide
3-[(3R,4S)-4-(morpholin-4-yl)-1-(1-phenyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]propan-1-ol
4-cyclobutyl-N-(1,4-dioxan-2-ylmethyl)-N,6-dimethylpyrimidin-2-amine
2-methyl-1-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1,4-diazepan-5-one
1-(cyclohexylmethyl)-5-{4-[(2-oxopyrrolidin-1-yl)methyl]piperidine-1-carbonyl}piperidin-2-one
3-(diphenylmethyl)-5-(pyrrolidin-1-ylmethyl)-1,2,4-oxadiazole
N4-[3-(1,3-benzothiazol-2-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
1-[(4aS,8aR)-1-[3-(dimethylamino)benzoyl]-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]ethan-1-one
1-(2-cyclohexylethyl)-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N,N-dimethyl-2-({1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidin-3-yl}formamido)acetamide
N-(2,2-dimethyloxan-4-yl)-2-ethyl-6-methyl-4-oxo-1-[2-(piperidin-1-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
5-ethyl-N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)pyrazolo[1,5-a]pyrimidin-7-amine
2-ethoxy-5-{2-[methyl(1,2-oxazol-3-ylmethyl)amino]pyrimidin-4-yl}benzoic acid
N-cyclopropyl-1-(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidin-4-yl)piperidine-3-carboxamide
N-[(2S)-3-(1H-imidazol-4-yl)-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-1-oxopropan-2-yl]acetamide