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methyl 3-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-1-(3-methylbutyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
N-{1-[(4-fluorophenyl)methyl]-7-(thiomorpholine-4-carbonyl)-1H-1,3-benzodiazol-5-yl}-2-methoxyacetamide
1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-[2-(1H-pyrrol-1-yl)ethyl]piperazine
(3S,5S)-1-[(3-methylthiophen-2-yl)methyl]-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
N-ethyl-6-(4-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperazin-1-yl)pyridine-3-carboxamide
(3S,4R)-1-[1-(4-methylphenyl)cyclopropanecarbonyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-3-(propan-2-yl)-N-(pyridin-3-ylmethyl)-1,2-oxazole-5-carboxamide
(2S,4R)-4-amino-1-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-N,N-diethylpyrrolidine-2-carboxamide
7-(4-methylphenyl)-4-[(3-methylpyridin-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{5-[(3-fluoro-2,4-dimethylphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1-propyl-1H-imidazole
N-{[2-(diethylamino)pyridin-3-yl]methyl}oxolane-3-carboxamide
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-2-(pyrimidin-2-ylsulfanyl)acetamide
N-[(3S,5S)-5-{[3-(1H-imidazol-1-yl)propyl]carbamoyl}-1-methylpyrrolidin-3-yl]morpholine-4-carboxamide
(3S,4S)-1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-4-propylpyrrolidine-3-carboxylic acid
(1S,5R)-6-propyl-3-[3-(trifluoromethyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-methyl-N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-1,3-thiazole-4-carboxamide
N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)(methyl)[2-(pyridin-2-yl)ethyl]amine
N-(1-ethyl-1H-1,2,4-triazol-3-yl)-3-(4-fluorophenyl)pyrrolidine-1-carboxamide
3-{2-oxo-2-[6-oxo-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-2-yl]ethyl}imidazolidine-2,4-dione
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]-5-methylpyrazine-2-carboxamide
(2S,4R)-4-amino-1-(2,3-dihydro-1H-indene-2-carbonyl)-N-methylpyrrolidine-2-carboxamide
(2S,4R)-4-amino-1-(2,3-difluoro-4-methoxybenzoyl)-N-ethylpyrrolidine-2-carboxamide
1-[1-(1-methylcyclopropanecarbonyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
(4aS,7aR)-1-[(3-fluoro-2,4-dimethylphenyl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-4-methylpentanamide
2-(ethoxymethyl)-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-{2-[(3-methoxyphenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}propanamide
3-{1-[3-(2-oxopyrrolidin-1-yl)propanoyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-5-methylthiophene-2-carboxamide
{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(2-methoxyethyl)(propan-2-yl)amine
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
{4-[(1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}pyrrolidin-3-yl)methyl]phenyl}methanol
1-(azepan-1-yl)-4-[4-(2-methylphenyl)-3-oxopiperazin-1-yl]butane-1,4-dione
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}ethan-1-one
ethyl 4-{1-[(4-chlorophenyl)methyl]-6-oxopiperidine-3-carbonyl}piperazine-1-carboxylate
2-amino-4-(2,3-dihydro-1,4-benzodioxin-6-yl)-6-(pyridin-2-yl)pyridine-3-carbonitrile
(3aS,6aR)-3-[(3,4-dimethoxyphenyl)methyl]-5-[(6-methylpyridin-2-yl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-(4-methanesulfonylphenyl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}acetamide
2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}acetamide
[(4-ethylphenyl)methyl]({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)amine
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
3-[(propan-2-yl)sulfamoyl]-5-(pyridin-4-yl)benzoic acid
2-[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]-N-(1-methyl-1H-pyrazol-4-yl)acetamide
1-(furan-2-carbonyl)-3-[2-(2-methylphenyl)ethyl]piperidine
3-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-1-(2-fluoro-5-methanesulfonamidophenyl)-3-methylurea
1-(3-methoxypropyl)-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione