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3-(5-{[3-(4-methylphenoxy)azetidin-1-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
1-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-8-yl)-3-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}urea
4-methanesulfonyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}benzamide
1-(furan-2-carbonyl)-3-{2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}piperidine
methyl 1-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}piperidine-4-carboxylate
2-(3-methoxyphenoxy)-1-[3-(2-methylpropyl)pyrrolidin-1-yl]ethan-1-one
6-chloro-2-{[(1R,5S,8R)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]methyl}quinoline
N-(1-hydroxybutan-2-yl)-5-(3-methoxyphenyl)-N-(pyridin-3-ylmethyl)furan-2-carboxamide
3-{4-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-1λ6-thiolane-1,1-dione
N2,N2,N4-trimethyl-N4-[(1-methyl-1H-imidazol-2-yl)methyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
7-(cyclopropylmethyl)-2-(3-ethoxypropanoyl)-2,7-diazaspiro[4.5]decan-6-one
5-cyclohexaneamido-N-(furan-2-ylmethyl)-1-(2-methoxyethyl)-1H-1,3-benzodiazole-7-carboxamide
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]propan-1-one
N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-[4-(4-ethylpiperazin-1-yl)piperidin-1-yl]-4-(1-methyl-1H-pyrazol-4-yl)pyrimidine
2-(3-phenylpropyl)-8-(pyrazin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
N-(1,3-dihydroxypropan-2-yl)-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-benzyl-4-(1H-imidazole-2-carbonyl)-1,4-diazepane-6-carboxylic acid
3-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1-{4-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}urea
4-(1H-1,3-benzodiazol-1-yl)-1-[2-(diethylamino)acetyl]piperidine-4-carboxylic acid
7-(3-chlorothiophene-2-carbonyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
9-[2-(benzyloxy)acetyl]-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(pyrrolidine-1-sulfonyl)ethyl]-2-(2,3,6-trimethylphenoxy)acetamide
1-(2-aminoethyl)-N-[1-(3,5-dichlorophenyl)-2-hydroxyethyl]-1H-1,2,3-triazole-4-carboxamide
(2R,6S)-4-[1-(3-chloropyridin-2-yl)piperidin-4-yl]-2,6-dimethylmorpholine
(3S,9aR)-3-[(4-hydroxyphenyl)methyl]-8-(thiophen-2-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-(4-methylpiperidin-1-yl)-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
[1-({[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]amino}methyl)cyclopentyl]methanol
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(2H-1,3-benzodioxol-5-yl)ethan-1-one
N-[(3R,4S)-4-cyclopropyl-1-methanesulfonylpyrrolidin-3-yl]-3-(6-oxo-1,6-dihydropyridazin-3-yl)propanamide
2-(adamantan-1-yl)-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]acetamide
4-{4-[(2-chloro-6-fluorophenyl)methyl]piperazin-1-yl}-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
3-[3-(2-methylphenyl)piperidine-1-carbonyl]-2-(methylsulfanyl)pyridine
4-{3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]pyridin-2-yl}morpholine
ethyl 3-{2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]acetamido}propanoate
3-(3-hydroxy-3-methylbutyl)-N-[3-(pyridin-2-yl)propyl]benzamide
N-{[3-(methylsulfanyl)phenyl]methyl}-2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
1-(2-methoxyethyl)-8-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(4-methoxyphenyl)methyl]-1-methyl-8-[4-(1H-pyrazol-1-yl)butan-2-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-({[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}amino)-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
N,1-dimethyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H-indole-6-carboxamide
8-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-methyl-3-(propan-2-yl)-5-(2,4,5-trifluorophenyl)-1H,4H-pyrazolo[3,4-d]imidazole
2-{3-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]phenoxy}acetamide
1-[(4-fluorophenyl)methyl]-N-methyl-N-[1-(pyridin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(3S,9aR)-3-benzyl-8-(4-chlorobenzenesulfonyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(4aR,8aS)-1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-6-(2-phenylethyl)-decahydro-1,6-naphthyridine
(4aS,8aR)-6-[(4-methyl-1H-imidazol-5-yl)methyl]-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
3-fluoro-N-methyl-N-{2-[4-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]ethyl}benzamide
4-methyl-2-[3-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]pyrimidine