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1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
3-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]-1-[4-(oxolan-2-ylmethoxy)phenyl]urea
1-[3-(1,3-oxazol-5-yl)phenyl]-3-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]urea
2-(2H-1,3-benzodioxol-5-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
N-(2-methoxyphenyl)-6-[(2-phenyl-1,3-thiazol-5-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
2-{4-[(3,5-difluorophenyl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
1-ethyl-3-methyl-N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)piperidine-3-carboxamide
(2,3-dihydro-1-benzofuran-5-ylmethyl)(ethyl){[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}amine
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-5-ethylpyrimidin-2-amine
N-[(3S,4R)-4-(4-methylphenyl)-1-[3-(methylsulfanyl)propyl]pyrrolidin-3-yl]acetamide
2-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-2,8-diazaspiro[4.5]decane
(3aR,6aS)-2-(cyclopropylmethyl)-5-(dimethyl-1,2-oxazole-4-carbonyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(3R,4S)-1-(cyclobutylmethyl)-4-propylpyrrolidin-3-yl]-2-(1H-1,2,3-triazol-1-yl)acetamide
(3R)-1-{[2-(5-methylfuran-2-yl)phenyl]methyl}pyrrolidin-3-ol
2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}acetamide
(1S,5R)-3-[2-(3-fluoro-4-hydroxyphenyl)acetyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(3-methoxyphenyl)methyl]-3-{1-[2-(phenylsulfanyl)acetyl]piperidin-3-yl}propanamide
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-(4,5-dimethyl-1H-imidazol-1-yl)ethan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-(methoxymethyl)-N-(pyridin-4-ylmethyl)furan-2-carboxamide
N-[3-hydroxy-1-(4-methylphenyl)propyl]-2,5-dimethyl-1,3-thiazole-4-carboxamide
3-{[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]methyl}pyridin-2-amine
1-{[2-(adamantan-1-yl)-1,3-thiazol-4-yl]methyl}-3-(hydroxymethyl)piperidin-3-ol
1-(3,4-dimethoxyphenyl)-2-[1-ethyl-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]ethan-1-amine
ethyl 4-[(4-chlorophenyl)methyl]-1-[3-(pyridin-3-yl)propanoyl]piperidine-4-carboxylate
{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
4-(5-methoxy-1H-indole-2-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(4-methylphenyl)methyl]acetamide
1-[2-(dimethylamino)-2-(3-methylphenyl)acetamido]-N-methylcyclohexane-1-carboxamide
{2-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]-1-(3-methylthiophen-2-yl)ethyl}dimethylamine
3-[3-(2-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
2-{1-[(3-hydroxyphenyl)methyl]piperidin-2-yl}acetamide
8-(cyclobutylmethyl)-2-[(3,5-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-chloro-5-acetamido-N,N-bis(pyridin-3-ylmethyl)benzamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-(2-methoxyacetamido)benzamide
3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}propan-1-one
N-[(3-hydroxypyrrolidin-3-yl)methyl]-2,3,4-trimethoxybenzamide
2-{4-[(4-methoxyphenyl)methyl]-3-oxopiperazine-1-carbonyl}pyrrolidine-1-carboxamide
2-(2-aminoethyl)-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]quinazolin-4-amine
2-({1-[(5-chloro-2,4-dimethoxyphenyl)methyl]piperidin-4-yl}oxy)pyrimidine
1-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-5-(1-methyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazole
1-{2-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]-2-oxoethyl}azepan-2-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(2-oxopyrrolidin-1-yl)butanamide
1-(1H-1,3-benzodiazole-5-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-(1-{[2-(propylamino)pyrimidin-5-yl]methyl}piperidin-3-yl)pyrrolidin-2-one
3-(3-methylbutyl)-2-oxo-1-[2-(1H-pyrrol-1-yl)ethyl]-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
{[4-methoxy-3-(methoxymethyl)phenyl]methyl}(methyl)[(3-methyl-1H-pyrazol-4-yl)methyl]amine
N-(2,3-dimethylphenyl)-5-[1-(1,2-oxazole-3-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
8-(4-methylpyrimidine-5-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
{1-[1-(2-fluorophenyl)cyclopropanecarbonyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
N-[4-(furan-2-yl)butan-2-yl]-2,4-dimethylpyrimidine-5-carboxamide