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1-({[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]carbamoyl}methyl)piperidine-4-carboxamide
(3S,4S)-1-(3-fluoropyridine-2-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
(2S,4R)-1-[(2,5-dimethylphenyl)methyl]-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
ethyl 1-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
2-(cyclopropylmethyl)-8-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-2,8-diazaspiro[5.5]undecan-3-one
N-[1-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]oxolane-3-carboxamide
N-(isoquinolin-5-ylmethyl)-N-methyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-[(5-methylfuran-2-yl)methyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
(3S,4S)-4-methyl-1-[(4-methyl-6-phenylpyrimidin-2-yl)methyl]piperidine-3,4-diol
(4aS,8aR)-6-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-1-(3-methylbutyl)-decahydro-1,6-naphthyridin-2-one
2-methoxy-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)butanamide
1-(cyclopropylmethyl)-5-({[4-(3-fluorophenyl)oxan-4-yl]methyl}amino)azepan-2-one
1-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-(pyrrolidin-1-yl)piperidine
1-{2-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-2-oxoethyl}-1,2,3,4-tetrahydroquinolin-2-one
3-hydroxy-5-(8-methylquinolin-5-yl)benzoic acid
3-ethyl-1-[4-(4-methylpiperazin-1-yl)benzoyl]piperidine-3-carboxylic acid
2-cyclopropyl-4-methyl-5-[2-(2-phenylethyl)piperidine-1-carbonyl]pyrimidine
2-(2-methanesulfonylethyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
6-(4-cyclopentyl-1,4-diazepan-1-yl)pyridine-2-carboxylic acid
4-(4-cyclobutanecarbonyl-1,4-diazepane-1-carbonyl)-N-methylpyridin-2-amine
2-methoxy-1-(4-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,4-diazepan-1-yl)ethan-1-one
(4-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-1,4-oxazepan-6-yl)methanol
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
2-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
2-[1-(2-methyl-1,3-benzothiazol-6-yl)-5-[2-(1H-pyrazol-1-yl)ethyl]-1H-1,2,4-triazol-3-yl]acetamide
1-{4-[(2-methylphenyl)methyl]piperazin-1-yl}-4-(1H-pyrazol-4-yl)butan-1-one
1-[(4-methyl-1H-imidazol-5-yl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
2-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-5-(1H-1,2,3,4-tetrazol-1-yl)phenol
4-(3-{[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]oxy}benzoyl)morpholine
1-{2-methyl-4-[4-(2-propoxyethyl)piperazin-1-yl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)benzenesulfonamide
(1S,6R)-9-(3-fluoropyridin-2-yl)-3,9-diazabicyclo[4.2.1]nonan-4-one
1-methyl-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-1H-pyrazole-5-carboxamide
[(3aS,6aS)-2-(3-propyl-1H-pyrazole-5-carbonyl)-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
1-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(pyridin-3-ylmethyl)piperazine
N-tert-butyl-4-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]morpholine-2-carboxamide
N-methyl-2-(3-methyl-1,2-oxazol-5-yl)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
6-methyl-2-({[3-(1H-1,2,4-triazol-1-yl)propyl]amino}methyl)quinolin-4-ol
6-[(3S,5R)-3-(hydroxymethyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-1-yl]pyridine-2-carbonitrile
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}cyclohex-3-ene-1-carboxamide
2,8-dimethyl-4-{4-[2-(1H-pyrrol-1-yl)ethyl]piperazine-1-carbonyl}quinoline
1-(3-chloro-2-propoxyphenyl)-3-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)urea
2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]-N-(3-phenylpropyl)acetamide
1-(2-methylphenyl)-4-{2-[(4-methylphenyl)methyl]benzoyl}piperazin-2-one
(2S)-3-(3,3-diphenylpiperidin-1-yl)-2-methylpropan-1-ol
3-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-1-{1-oxaspiro[4.4]nonan-3-yl}urea
4-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]quinoline
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,2-oxazole-3-carboxamide
1-[1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-3-phenylpropan-1-one