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N-(butan-2-yl)-1-cyclopentyl-4-oxo-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1,4-dihydropyridine-3-carboxamide
5-{[5-(1-acetamidoethyl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}-N-methylfuran-2-carboxamide
2-{1-[(3-methoxyphenyl)methyl]-4-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
methyl 3-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-7-oxo-9-(thiophen-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}phenyl)-1H-imidazole
methyl 5-(3-acetamidothiophene-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-[1'-(3-ethyl-1,2-oxazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
3-methyl-8-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(pyridin-3-ylmethyl)-1-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
3-({2-[(thiophen-2-ylmethyl)amino]phenyl}formamido)propanamide
2-methyl-3-{[1-(3-methylbutyl)-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}quinoxaline
N-(hexahydro-1H-pyrrolizin-7a-ylmethyl)-3-(3-hydroxy-3-methylbutyl)benzamide
3-{5-[2-(1H-pyrrol-1-yl)propan-2-yl]-1,2,4-oxadiazol-3-yl}pyridazine
7-(2,3-dimethoxyphenyl)-9-methoxy-4-{[4-(propan-2-yl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-(1H-indol-1-ylmethyl)-N-methyl-N-[(1-methylpiperidin-2-yl)methyl]-1H-pyrazole-3-carboxamide
2-[({5-[1-(4-methoxypyrimidin-2-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
3-[1-(1-aminocyclopropanecarbonyl)piperidin-3-yl]-1-[2-(dimethylamino)ethyl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
8-(3-fluoropyridin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-cyclopentanecarbonyl-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}piperidine-4-carboxamide
2-methyl-5-phenyl-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[1-(2-phenylethyl)piperidin-3-yl]-1H-indole-5-carboxamide
3-(2-methoxyethyl)-5-[1-methyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]-1,2,4-oxadiazole
3-methyl-N-{1-[1-(2-methylpyrimidin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetamide
5-{2-azaspiro[4.4]nonane-2-carbonyl}thiophene-2-carboxylic acid
N-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}-2,2-dimethyloxane-4-carboxamide
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
1-[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one
3-[2-(1H-pyrazol-1-ylmethyl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{3-[4-(1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyrimidine
N-[(4-methylphenyl)(thiophen-2-yl)methyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
methyl 2-[3-(1H-imidazol-1-yl)propyl]-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
2-[2-(dimethylamino)ethyl]-9-(2-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
ethyl 5-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-{[4-(3-methylpyridin-4-yl)phenyl]methyl}methanesulfonamide
4-[2-(2-ethoxyphenyl)-1H-imidazol-1-yl]-1-(2-methoxyethyl)pyrrolidin-2-one
6-(2-chlorophenyl)-2-(4-{[(2-hydroxyethyl)(methyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
6-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-indole
4-{2-[2-(propylsulfanyl)pyrimidin-5-yl]-1H-imidazol-1-yl}benzamide
[(3S,5R)-1-(4-fluoro-2-methylbenzoyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
4,4-difluoro-1-({2-[3-(1H-imidazol-1-yl)propoxy]-3-methoxyphenyl}methyl)piperidine
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-3-(1,2-oxazolidin-2-yl)propanamide
5-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-2-one
4-{[4-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-2,1,3-benzoxadiazole
7-(3,6-dimethylpyrazin-2-yl)-4-(2-fluorobenzoyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-methyl-N-({1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl}methyl)furan-2-carboxamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
butyl N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)carbamate
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl][2-(3-methoxyphenoxy)ethyl]methylamine