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4-({[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl](propan-2-yl)amino}methyl)-6,7-dimethyl-2H-chromen-2-one
N-benzyl-N-methyl{[(1S,2R)-2-aminocyclobutyl]amino}sulfonamide
N-{[(1R,2S,5R)-6,6-dimethylbicyclo[3.1.1]heptan-2-yl]methyl}-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
1-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-[ethyl(methyl)amino]propan-1-one
N-{3-[(5-methylpyridin-2-yl)amino]propyl}-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
5-[(dimethylamino)methyl]-N-[(4-fluorophenyl)methyl]-N-methyl-1,3,4-oxadiazole-2-carboxamide
6-tert-butyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4,6-dimethoxy-2-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}pyrimidine
1-(furan-3-carbonyl)-3-[3-(trifluoromethyl)benzoyl]piperidine
3-(2,5-dimethoxyphenyl)-1-(3-fluorobenzoyl)pyrrolidine
N-{[5-({4-[1-(dimethylamino)ethyl]piperidin-1-yl}methyl)furan-2-yl]methyl}-N-methylmethanesulfonamide
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-propyl-1H-pyrazole-5-carboxamide
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-3-(2-oxoimidazolidin-1-yl)benzamide
3-methyl-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}furan-2-carboxamide
4-{[methyl(oxolan-3-ylmethyl)carbamoyl]amino}-N-(2-phenylethyl)benzamide
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-2,8-dimethylquinoline-4-carboxamide
(2R,3R,6R)-3-(2-methoxyphenyl)-5-methyl-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{2-[(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)amino]pyrimidin-4-yl}piperidin-4-ol
2-(4-{[(3R)-3-hydroxypyrrolidin-1-yl]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
1-[(4-ethylphenyl)methyl]-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
1-(1,3-benzoxazol-2-yl)-N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-amine
3-[6-(dimethylamino)pyridazin-3-yl]-5-[2-(piperidin-2-yl)ethyl]phenol
N-(1-benzyl-1H-pyrazol-5-yl)-2-[3-(2-methylphenyl)-1H-pyrazol-1-yl]acetamide
4-({5-[1-(ethanesulfonyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
methyl 2-[methyl(2-phenylethyl)sulfamoyl]-6-(oxolane-2-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(1R,2S)-N1-butyl-N2-[(4,6-dimethylpyridin-3-yl)methyl]cyclohexane-1,2-dicarboxamide
2-{[ethyl(oxan-4-yl)amino]methyl}benzoic acid
1-(4-methanesulfonylphenyl)-3-[(3R)-pyrrolidin-3-yl]urea
3-(1,2,3,6-tetrahydropyridin-1-ylmethyl)-N-(1,2,3-thiadiazol-5-yl)benzamide
N-[3-(3-fluorophenyl)phenyl]-2-(morpholin-3-yl)acetamide
4,6-dimethyl-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
4-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-3,4-dihydro-2H-1,4-benzothiazin-3-one
4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)benzamide
8-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
8-(butan-2-yl)-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N3-cyclopentyl-N5-[2-(3-fluorophenyl)ethyl]-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
3-{1-[2-(3-hydroxyphenyl)acetyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
3-[2-(dimethylamino)ethyl]-8-(5-methoxy-4-oxo-4H-pyran-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-methoxy-N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
8-(6-carboxypyrazin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(2-aminoethyl)(methyl){[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}amine
N-[(2,3-dimethoxyphenyl)methyl]-5-methyl-N-(pyridin-3-ylmethyl)-1,3-oxazole-4-carboxamide
2-ethoxy-4-({3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenol
7-(oxane-4-carbonyl)-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}pyrimidin-4-amine
N-{[3-(cycloheptyloxy)-4-methoxyphenyl]methyl}-N-cyclopropyl-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
1-[2-(4-methoxyphenyl)ethyl]-N-(1-methylpiperidin-4-yl)-6-oxopiperidine-3-carboxamide
3-{5-[(2,6-difluoro-4-methoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
4-[5-(3-propyl-1H-pyrazole-5-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl]morpholine
N-[4-methoxy-2-(2-methylpropanamido)phenyl]-2-methylpentanamide