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8-[2-(2-hydroxyethoxy)ethyl]-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-(4-methoxybenzoyl)-4-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazine
6-{1-[(2-methyl-2H-indazol-3-yl)methyl]piperidin-3-yl}-3,4-dihydropyrimidin-4-one
5-(2-methoxy-5-methylphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-({[1-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
N-(2,4-dimethylphenyl)-2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3,4-dimethyl-5-sulfamoylbenzamide
5-ethyl-N-(quinolin-3-ylmethyl)pyrimidin-2-amine
1'-(1-benzofuran-5-ylmethyl)-5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(4-ethoxyphenyl)methyl]-N-(2-methoxyethyl)-1-methyl-1H-pyrrole-2-carboxamide
methyl 4-[5-({ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-1,2,4-oxadiazol-3-yl]benzoate
N-[3-(2-methylphenyl)phenyl]-4-(morpholin-4-yl)piperidine-1-carboxamide
5-[3-(cyclopentyloxy)phenyl]-1-methyl-1H,4H-pyrazolo[3,4-d]imidazole
1-[(1-phenylcyclohexyl)methyl]piperidin-4-ol
N-ethyl-2-hydroxy-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)acetamide
N-(1-benzothiophen-2-ylmethyl)-6-{[ethyl(2-methylprop-2-en-1-yl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(1-{5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridin-2-yl}piperidin-4-yl)ethan-1-ol
ethyl 3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
1-[2-({[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]amino}methyl)morpholin-4-yl]ethan-1-one
1-(dimethyl-1,2-oxazole-4-carbonyl)-3-(4-methylphenoxymethyl)piperidine
N-[(3S,4R)-1-[(2,4-difluorophenyl)methyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
N-[(2R,3R)-2-methoxy-1'-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
4-[3-(azocan-1-yl)propanamido]butanoic acid
N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)-2-oxo-2-phenylacetamide
5-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}-4-methyl-1H-imidazole
1-{3-[5-(2-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl}-4,4,4-trifluorobutan-1-one
8-(furan-3-ylmethyl)-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-benzyl-3-{2-[3-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
1-(6-chloro-1,3-benzothiazol-2-yl)-N-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidin-4-amine
1-(azepan-1-yl)-3-[(5-ethyl-2-methylpyrimidin-4-yl)amino]propan-2-ol
2-{2-[(4-hydroxyazepan-1-yl)methyl]-4-(pyridin-2-yl)phenoxy}acetic acid
6-chloro-3-(1H-imidazol-2-yl)-N,N-dimethylimidazo[1,2-a]pyridine-2-carboxamide
3-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,6-dichlorophenyl)urea
5-(2-{4-[(3-fluorophenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)-2,6-dimethyl-3,4-dihydropyrimidin-4-one
1-(azepan-1-yl)-3-[3-({[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
3-[4-oxo-7-(trifluoromethyl)-3,4-dihydroquinazolin-3-yl]propanamide
N-[2-(1H-pyrazol-4-yl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
6-{[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]amino}-N,N-dimethylpyrazine-2-carboxamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
N-[3-(2,4-dimethylphenoxy)propyl]-N,1-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(2,3-dihydro-1-benzofuran-7-carbonyl)-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
2,6-dimethyl-N-[1-(pyridin-4-yl)propan-2-yl]quinoline-3-carboxamide
(3S,4S)-N-(adamantan-1-yl)-3,4-dihydroxypiperidine-1-carboxamide
5-methyl-N-(5-oxo-1-phenylpyrrolidin-3-yl)-3-phenyl-1,2-oxazole-4-carboxamide
7-chloro-4-[3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]quinoline
N-ethyl-N-(2-methylphenyl)-3-[4-(oxan-4-yl)piperazin-1-yl]propanamide
3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-6-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
3-[(3R,4S)-1-(1H-indole-6-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
2,4-dimethyl-6-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyrimidine