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N-[(3S)-1-[2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]pyrrolidin-3-yl]acetamide
N-(3-fluorophenyl)-3-({[4-(pyrrolidine-1-carbonyl)phenyl]methyl}amino)propanamide
N-(1-ethyl-5-oxopyrrolidin-3-yl)-2,6-dimethylquinoline-4-carboxamide
2-({[1-(3,4-dimethoxybenzoyl)piperidin-3-yl]oxy}methyl)pyridine
3-({2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}methyl)pyridin-2-amine
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-({[(4-hydroxy-1-methylpiperidin-4-yl)methyl]amino}methyl)piperidin-2-one
6-cyclopentyl-N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(1S,5R)-6-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
methyl({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)(quinolin-8-ylmethyl)amine
2-cyclopropyl-N-{[4-(3-methylpiperidin-1-yl)phenyl]methyl}-6-oxo-1,6-dihydropyrimidine-5-carboxamide
N-methyl-1-[(7-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperidine-3-carboxamide
6-methyl-2-oxo-N-(3-phenylprop-2-yn-1-yl)-N-propyl-1,2-dihydropyridine-4-carboxamide
1-{1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]piperidin-4-yl}piperidin-4-ol
1-(oxan-4-yl)-4-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}piperazine
8-[(5-methylpyrazin-2-yl)methyl]-9-oxo-N-propyl-2,8-diazaspiro[5.5]undecane-2-carboxamide
2-{[(5-ethylpyridin-2-yl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1H-indole-5-carboxamide
8-(7-chloroquinoxalin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
3-(cyclohexylamino)-N,N-dimethylazepane-1-sulfonamide
1-[2-(dimethylamino)ethyl]-3-(1H-indazol-5-yl)-1-[(5-methylthiophen-2-yl)methyl]urea
(4aR,7aS)-1-(2-hydroxyethyl)-4-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-methoxy-N-(2-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
[(3-chloro-4-methoxyphenyl)methyl](oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amine
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(4-methoxyphenyl)acetamide
N-[(3R,4R)-3-hydroxy-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl]pyrazine-2-carboxamide
3-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-N-(3-methoxyphenyl)propanamide
2-amino-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]pyridine-4-carboxamide
2-(4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl}-1H-1,2,3-triazol-1-yl)ethan-1-amine
2-{4-[7-fluoro-4-(thiomorpholine-4-carbonyl)quinolin-2-yl]-1H-pyrazol-1-yl}ethan-1-ol
6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-4-(pyrazine-2-carbonyl)-1,4-diazepan-2-one
(3R,4R)-N-(cyclohexylmethyl)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidine-1-carboxamide
6-(1-methyl-1H-imidazol-2-yl)-N-[1-(thiophen-3-yl)propan-2-yl]pyridazin-3-amine
1-{2-[4-(4-methylphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
4-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylquinoline
9-(3-hydroxy-4-methoxybenzoyl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(2,6-difluoro-3-methoxyphenyl)methyl]-N-methyloxan-4-amine
(3S,4S)-1-(4-methoxybenzoyl)-4-({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)pyrrolidin-3-ol
3-[1-({4-[methyl(phenyl)amino]phenyl}methyl)piperidin-3-yl]propan-1-ol
1-[2-(dimethylamino)-4-(4-hydroxypiperidin-1-yl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]-2-(methylsulfanyl)ethan-1-one
(1S,5R)-3-methyl-6-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-3,6-diazabicyclo[3.2.2]nonane
ethyl 4-[3-(4-methyl-1,3-thiazol-5-yl)propanamido]piperidine-1-carboxylate
N-[(5-methylfuran-2-yl)methyl]-2-[2-(1H-pyrazol-1-yl)acetyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
2-(1-{3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}piperidin-4-yl)-1,2,3,4-tetrahydroisoquinoline
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[2-(6-hydroxypyrimidin-4-yl)ethyl]propanamide
3-{4-oxo-3H,4H-pyrido[3,4-d]pyrimidin-3-yl}azepan-2-one
3-({1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-yl}amino)-2,3-dihydro-1λ6-thiophene-1,1-dione
1-{[5-(cyclohexylsulfanyl)furan-2-yl]methyl}-N-methylpyrrolidine-3-carboxamide
N-{[5-(4-fluorophenyl)furan-2-yl]methyl}-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]acetamide