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(4aS,8aR)-6-(furan-2-ylmethyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-2-(2-methylphenyl)pyrrolidine
6-methyl-2-oxo-N-[3-(pyridin-4-yl)propyl]-1,2-dihydropyridine-4-carboxamide
5-(morpholin-4-ylmethyl)-N-(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)furan-3-carboxamide
N-benzyl-5-{[3-(morpholin-4-yl)azetidin-1-yl]methyl}pyrimidin-2-amine
N-(furan-2-ylmethyl)-9-methoxy-7-oxo-3-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-(1-cyclohexyl-2,6,6-trimethyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-[2-(dimethylamino)ethyl]acetamide
1-{6-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]pyridin-2-yl}ethan-1-ol
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
1-{[1-ethyl-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
9-[(2-chlorophenyl)methyl]-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(2-amino-1,3-thiazol-4-yl)methyl]-2-(azepan-1-yl)acetamide
(1R,5R)-N,N-dimethyl-6-(3-propyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-(2-fluorophenyl)-5-[(pyridin-2-ylmethyl)sulfamoyl]benzoic acid
4-ethyl-5-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}-1-methyl-1H-pyrazole-5-carboxamide
3-{[(2-ethyl-1,3-dihydroxypropan-2-yl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-[4-(3,4-dichlorophenyl)piperazin-1-yl]-2-(oxolan-2-ylmethoxy)ethan-1-one
[2-(1H-imidazol-1-yl)ethyl]({[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl})methylamine
N-cyclooctyl-2-{[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]amino}acetamide
2-(1,3-benzoxazol-2-yl)-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]acetamide
N-methyl-N-[2-(pyridin-2-yl)ethyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carboxamide
2-(3-hydroxypiperidin-1-yl)-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]acetamide
4-{4-[4-(furan-2-carbonyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-[2-(4-fluorophenyl)ethyl]-N-{[2-(3-hydroxypiperidin-1-yl)-5,8-dimethoxyquinolin-3-yl]methyl}-1,3-thiazole-5-carboxamide
N-[(2S)-1-hydroxypropan-2-yl]-4-{[2-(1H-pyrrol-1-yl)ethyl]sulfamoyl}benzamide
1-benzyl-5-[1-(4-chloro-1H-pyrazol-1-yl)ethyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
1-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
(3R,4R)-4-cyclopropyl-3-methyl-1-[(2,3,5,6-tetrafluoro-4-methoxyphenyl)methyl]piperidin-4-ol
3-(2H-1,3-benzodioxol-5-yl)-5-[(5-chlorothiophen-2-yl)methyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
{2-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-1,3-thiazol-4-yl}methanol
3-{5-[(8-methoxy-2H-chromen-3-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
methyl 5-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
2-[1-(1,3-thiazol-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
5-{3-cyclopentyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-4-methyl-1H-imidazole
4-methylphenyl (7R,9aR)-7-(2-methylpropyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
(1S,5R)-6-(cyclobutylmethyl)-3-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-2-methylpyrido[2,3-d]pyrimidin-4-amine
2-[(3,5-difluorophenyl)methyl]-8-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-(1-benzothiophen-3-yl)-2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}acetic acid
2-(2-{[3-methyl-4-(propan-2-yl)piperazin-1-yl]methyl}phenoxy)ethan-1-ol
1-(2-methyl-4-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
2-(prop-2-en-1-yl)-9-{spiro[2.3]hexane-1-carbonyl}-2,9-diazaspiro[5.5]undecan-3-one
N,N-dimethyl-2-[(1S,5R)-3-(2-methylquinolin-4-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
4-[1-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1H-imidazol-2-yl]-2,1,3-benzoxadiazole
6-(3-acetamidophenyl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
1-(5-chloro-2-methylphenyl)-4-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}piperazine
1-{3-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
7-(oxan-4-yl)-N-[(2R)-oxolan-2-ylmethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-ethyl-5-[(4-methanesulfonylphenyl)methyl]-3-(phenoxymethyl)-1H-1,2,4-triazole