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methyl 3-(2H-1,3-benzodioxole-5-carbonyl)-7-oxo-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}pyridin-2-amine
3-methoxy-1-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}propan-1-one
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(4-fluorophenyl)ethan-1-one
(3aR,6aS)-5-{5-[(dimethylamino)methyl]furan-2-carbonyl}-2-ethyl-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[1-(4-propylphenyl)-1H-pyrazol-4-yl]ethan-1-ol
4-(2-{[3-oxo-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]amino}ethyl)benzene-1-sulfonamide
5-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]-N,N,4-trimethylpyrimidin-2-amine
2-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidin-4-amine
{4-[(2-chlorophenyl)methyl]-1-(oxane-4-carbonyl)piperidin-4-yl}methanol
(4aR,7aS)-1-methyl-4-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{5-cyclopropyl-4-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}-4-(2-fluorophenyl)pyrimidine
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyrimidin-4-ylmethyl)acetamide
N-[(3R,4R)-3-hydroxy-1-(4-sulfamoylbutanoyl)piperidin-4-yl]pyridine-3-carboxamide
(benzylsulfamoyl)({2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl})amine
2-(1-methyl-4-{[4-(2-methylphenyl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
1-cyclopropyl-N-{[5-(4-fluorophenyl)furan-2-yl]methyl}-5-oxopyrrolidine-3-carboxamide
4-{1-[(3-methoxyphenyl)methyl]-6-oxopiperidine-3-carbonyl}piperazin-2-one
1-(2-amino-6-methylpyrimidin-4-yl)-4-(pyridin-2-yl)piperidin-4-ol
N-{1-[(2-fluoro-4-methoxyphenyl)methyl]azepan-3-yl}-2-(thiophen-2-yl)acetamide
1-(2-methoxybenzoyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-[(5-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-2-methoxyphenyl)methyl]-1H-1,2,4-triazole
1-{[2-(benzyloxy)phenyl]methyl}-N-methylpiperidine-2-carboxamide
4-[2-amino-6-(cyclopropylamino)pyrimidin-4-yl]-1-[(4-fluorophenyl)methyl]piperazin-2-one
4-methyl-N-(quinolin-5-yl)-1,4-diazepane-1-carboxamide
N3-cyclopentyl-N5-[1-(furan-2-yl)ethyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
5-{2-[3-(morpholine-4-carbonyl)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-oxo-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
2-[(1-cyclopropanecarbonylpiperidin-4-yl)formamido]-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetic acid
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyridazine-3-carboxamide
N-benzyl-N-(3-methylbutan-2-yl)-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
3-[methyl({[2-(1H-pyrazol-1-yl)phenyl]methyl})amino]propane-1,2-diol
N-{[3-methyl-7-(5-propyl-1,2-oxazole-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-phenoxypropanamide
N-[(3,4,5-trimethoxyphenyl)methyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
3-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-1-(1H-indazol-7-yl)-3-methylurea
(2S,4S)-4-amino-N-benzyl-1-methyl-N-[(6-methylpyridin-2-yl)methyl]pyrrolidine-2-carboxamide
1-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-3-(1-propyl-1H-1,3-benzodiazol-5-yl)urea
1-{1-[(dimethyl-1,3-thiazol-2-yl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-N,N-bis(prop-2-en-1-yl)acetamide
6-methyl-2-[1-(pyridazine-3-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
N-[4-(furan-2-yl)butan-2-yl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
N-[2-(3-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenoxy)propyl]imidazo[1,2-a]pyridine-2-carboxamide
N-{1-[1-(pent-4-enoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
4-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(4-fluorophenyl)methyl]piperazin-2-one
3-methyl-3-phenyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]butanamide
dimethyl(2-{2-[1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
4-cyclobutyl-2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-methylpyrimidine
5-(1,1-dioxo-1λ6-thiomorpholine-4-carbonyl)-2,3-dimethylbenzene-1-sulfonamide
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-3-(1H-pyrazol-1-yl)benzamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol