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4-[(5-{[(dimethyl-1,2-oxazol-4-yl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
6-{3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]propanoyl}-2-(2-hydroxyethyl)-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3-(3,5-dimethyl-1H-pyrazol-4-yl)propanamide
4-{4-[2-(dimethylamino)-2-(4-fluorophenyl)acetyl]piperazin-1-yl}benzonitrile
1-[2-(1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)ethyl]pyrrolidin-2-one
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-ethyl-N-[2-(pyridin-2-yl)ethyl]piperidin-4-amine
2-(5-{[3-(2,6-dimethylphenoxy)azetidin-1-yl]methyl}furan-2-yl)benzonitrile
2-methoxy-1-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-cyclopropyl-4-methyl-N-{[3-(oxan-2-ylmethoxy)phenyl]methyl}benzamide
N-[2-(1H-pyrazol-1-yl)phenyl]-4-(thian-4-yl)piperazine-1-carboxamide
1-({2-[({1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]phenyl}methyl)pyrrolidin-2-one
(3R,4R)-4-(hydroxymethyl)-1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-3-ol
5-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-2-(3,4,5-trimethoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
1-methyl-3-[1-(1,2,5-oxadiazole-3-carbonyl)piperidin-4-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-({4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-4-methoxypyridine
4-{4-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]piperidin-1-yl}-6-methyl-2-phenylpyrimidine
3-[(3R,4S)-4-(dimethylamino)-1-[(2-fluoro-4-methylphenyl)methyl]piperidin-3-yl]propan-1-ol
1-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-5-methyl-5-phenylpiperidin-2-one
5-(2-chloro-4-methoxyphenoxymethyl)-N-methyl-N-(oxolan-3-yl)-1H-pyrazole-3-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-1-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}propan-1-one
7-[(2-fluorophenyl)methyl]-2-(oxan-4-yl)-2,7-diazaspiro[4.5]decane
3-{[1-(pyrimidin-2-yl)piperidin-4-yl]methyl}benzoic acid
methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]{[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
1-cyclopentyl-3-(4-phenylazepane-1-carbonyl)-5-(piperidine-1-carbonyl)-1,4-dihydropyridin-4-one
3-[2-(dimethylcarbamoyl)-4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl]piperidine-1-carboxamide
4-(2-hydroxy-3-methoxybenzoyl)-5-methyl-1-(3-methylphenyl)piperazin-2-one
2,5,6-trimethyl-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)pyrimidin-4-amine
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)propanamide
2-[3-(pyridin-4-yl)azetidin-1-yl]-5-(trifluoromethyl)pyridine
7-methyl-2-(pyrimidin-5-yl)-4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)quinoline
5-fluoro-N4,N4-dimethyl-N2-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]pyrimidine-2,4-diamine
1-[(4-chlorophenyl)methyl]-N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-{1-[1-(2-hydroxypropyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxybenzamide
5-methyl-N-{3-[2-(pyridin-4-yl)-1H-imidazol-1-yl]propyl}pyridin-2-amine
2-(4-methoxy-2,6-dimethylphenyl)-2-[4-(pyridin-2-ylmethyl)piperazin-1-yl]acetic acid
2-{1-benzyl-4-[(1-ethyl-1H-imidazol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-[(4aS,8aR)-2-oxo-1-propyl-decahydro-1,6-naphthyridin-6-yl]-N-cyclopropylpyridine-4-carboxamide
1-(2-{5-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-3-yl}ethyl)pyrrolidin-2-one
1-[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
5-chloro-2-methyl-4-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyrimidine
(1R,5S,6S)-3-[(2E)-2-methylbut-2-en-1-yl]-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-3-azabicyclo[3.1.0]hexane-6-carboxamide
N-(1H-imidazol-2-ylmethyl)-2-phenyl-5,6,7,8-tetrahydroquinazolin-5-amine
2-[({5-[1-(5-methoxyfuran-2-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
4-hydroxy-2-(pyridin-3-yl)-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]pyrimidine-5-carboxamide
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-[2-(methylsulfanyl)pyrimidin-4-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(3-butanamidophenyl)-4-(pyrrolidin-3-yl)piperazine-1-carboxamide
1-[4-(2-methoxybenzoyl)piperazin-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
5,6-dimethoxy-2-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1,2-dihydroisoquinolin-1-one