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N-ethyl-7-fluoro-2-(2-methylpyrimidin-5-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]quinoline-4-carboxamide
1-[3-(2-methylpropyl)pyrrolidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1H-1,2,3-triazole-5-carboxamide
1-[(3-fluorophenyl)methyl]-4-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperazine
2-ethyl-9-(1-methyl-1H-pyrazole-5-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
ethyl 1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
(2S)-2-amino-1-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
{4-[(4-methoxyphenyl)methyl]-1-(quinoline-6-carbonyl)piperidin-4-yl}methanol
6-[(diethylamino)methyl]-N-[2-(1H-imidazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-(4-methylpyrimidine-5-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
4-[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]-1-(3,5-dimethylphenyl)piperazin-2-one
2-[4-(3-phenylphenyl)-1H-pyrazol-1-yl]propanamide
2-(2-hydroxyphenyl)-1-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-amine
1-(2-methoxyphenyl)-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-1H-pyrazole-4-carboxamide
4-(7-methoxy-2-methylquinoline-4-carbonyl)-3,4-dihydro-2H-1,4-benzoxazine
(4aS,8aR)-6-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
5-cyclopropanecarbonyl-1'-(5-propyl-1,3,4-thiadiazol-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
6-methyl-2-[(2-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}ethyl)amino]-3,4-dihydropyrimidin-4-one
(furan-2-ylmethyl)(methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
methyl 4-(4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}piperidin-1-yl)-4-oxobutanoate
N-(4-fluorophenyl)-1-[3-(prop-2-en-1-yloxy)benzoyl]piperidin-3-amine
N-[2-(4-hydroxypiperidin-1-yl)-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl]-3-methylfuran-2-carboxamide
3-ethyl-8-(6-methyl-2-oxo-1,2-dihydroquinoline-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(pyridin-2-ylmethyl)-1-[1-(3,3,3-trifluoropropanoyl)piperidin-4-yl]piperidine-3-carboxamide
N-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(4-chlorophenoxy)pyridine-3-carboxamide
8-{[3-(difluoromethoxy)phenyl]methyl}-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
8-[4-amino-6-(benzylamino)-1,3,5-triazin-2-yl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(3S,4S)-1-[3-(dimethylamino)-1,2,4-thiadiazol-5-yl]-4-propylpyrrolidine-3-carboxylic acid
(2S,4S)-N-ethyl-1-methyl-4-[4-(piperidin-1-yl)benzamido]pyrrolidine-2-carboxamide
[(3R,4R)-1-(2,5-difluorobenzoyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
N-[(1R,2R)-2-acetamido-2,3-dihydro-1H-inden-1-yl]-1H-1,2,3-triazole-5-carboxamide
(1R,5R)-6-(2-methoxyethyl)-3-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
4-{[(3,6-dimethylpyrazin-2-yl)amino]methyl}-1λ6-thiane-1,1-dione
2-({2-[(1,2,3,4-tetrahydronaphthalen-1-yl)carbamoyl]phenyl}amino)acetic acid
N-[3-(1H-indazol-1-yl)propyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
2-amino-2-methyl-1-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propan-1-one
(1R,7S)-3-tert-butyl-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
3-(3-methylbut-2-en-1-yl)-1-(pyridin-4-ylmethyl)piperidine-3-carboxylic acid
methyl (2S)-2-{[1-(4-methylquinazolin-2-yl)pyrrolidin-2-yl]formamido}-2-phenylacetate
4-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-oxo-3,4-dihydroquinoxaline-2-carboxamide
N-[(2-fluorophenyl)methyl]-5-[(2-methoxyethyl)(methyl)amino]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(2,4-dimethoxy-3-methylphenyl)-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-5-methyl-1,3-oxazole
N-(3-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-3-oxopropyl)-N-methylmethanesulfonamide
N-[2-(3-fluorophenyl)ethyl]-2-[4-(4-{[1-(pyridin-3-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]acetamide
6-methyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
1-({2-cyclopropyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)-3-ethoxypropan-2-ol
[(1-cyclopentylpiperidin-4-yl)methyl][(2-fluoro-4-methoxyphenyl)methyl](pyridin-3-ylmethyl)amine
(2R,6S)-1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-2,6-dimethylpiperidine
N,N-dimethyl-6-[3-(1H-pyrazol-3-yl)phenyl]pyridazin-3-amine