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3-{1-[3-(1,2-oxazinan-2-yl)propanoyl]piperidin-4-yl}-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
2-{4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-N-(3-fluoro-2-methylphenyl)acetamide
N-[2-fluoro-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidine-1-carboxamide
4-{1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}-4-oxobutane-1-sulfonamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
2-(2-methoxyethyl)-8-[(5-propylfuran-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-1-phenylcyclopropane-1-carboxamide
1-[2-(1H-imidazol-5-yl)ethyl]-3-(oxan-4-yl)-5-(4,5,6,7-tetrahydro-2-benzothiophen-1-yl)-1H-1,2,4-triazole
5-{[2-(2-ethyl-1H-1,3-benzodiazol-1-yl)butanamido]methyl}-N-methylfuran-2-carboxamide
4-[(2-butyl-1H-imidazol-4-yl)methyl]-5-methyl-1-(3-methylphenyl)piperazin-2-one
2-(2,4-dichlorophenoxy)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]acetamide
N-[2-(dimethylamino)-2-(pyridin-2-yl)ethyl]-5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
5-(4-methyl-1,4-diazepan-1-yl)-2-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-2,3-dihydropyridazin-3-one
2-amino-8-(3,4-dimethylphenyl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
N-ethyl-4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-(pyridin-4-ylmethyl)butanamide
3-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-(thiophen-3-ylmethyl)benzamide
3-[(3R,4S)-1-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
N-{2-[3-(2H-1,3-benzodioxol-5-yl)propanamido]-5-methoxyphenyl}-2-methylpropanamide
N-[5-(oxolan-2-yl)-1,3,4-thiadiazol-2-yl]-2-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}acetamide
N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-3-(pyridin-3-yl)propanamide
(3S,4S)-1-(adamantan-1-yl)-4-(morpholin-4-yl)pyrrolidin-3-ol
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-5-methyl-1,2-oxazole-3-carboxamide
2-{[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]methyl}-6,8-dimethylquinolin-4-ol
N-(1,3-dimethyl-1H-pyrazol-5-yl)-1-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]piperidin-4-amine
4-methyl-3-({2-[(1S,5R)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamido}methyl)benzoic acid
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)cycloheptanecarboxamide
N,N-dimethyl-3-{methyl[1-(4-methylpyridin-2-yl)propan-2-yl]sulfamoyl}benzamide
(4aS,8aR)-6-[3-(dimethylamino)benzoyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1H-pyrazol-4-yl)propanamide
4-(cyclobutylsulfamoyl)-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]benzamide
1-(2-{1-[2-(morpholin-4-yl)benzoyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
2-[(4-chlorophenyl)methyl]-8-(3-fluoropropyl)-2,8-diazaspiro[4.5]decan-3-one
5-(2,6-dimethylpyrimidine-4-carbonyl)-N-ethyl-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-[(3R,4S)-3-(dimethylamino)-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-N,N-dimethylpropane-1-sulfonamide
4-(1-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}piperidin-4-yl)pyridine
2-[(5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-yl)amino]propane-1,3-diol
1-(4-methylphenyl)-4-[2-(3-methylphenyl)acetyl]piperazin-2-one
1-{4-[(butylsulfanyl)methyl]-5-methylfuran-2-carbonyl}-4-(1H-imidazol-2-yl)piperidine
2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]acetamide
4-chloro-N,N-diethyl-3-(2-methanesulfonylacetamido)benzamide
4-{[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]methyl}-1-methyl-1H-pyrrole-2-carbonitrile
5-methoxy-2-[3-(3-methylthiophene-2-carbonyl)piperidine-1-carbonyl]-1,4-dihydropyridin-4-one
6-{[2-(2-methoxyethyl)piperidin-1-yl]methyl}naphthalen-2-ol
2-(2,5-dimethoxyphenyl)-5-methyl-4-[(2-methyl-1H-imidazol-1-yl)methyl]-1,3-oxazole
8-{[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}quinoline
5-[1-(1,1-dioxo-1λ6-thiolan-3-yl)-3-phenyl-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-[2-(2-ethoxyethoxy)benzoyl]-1-(4-methylphenyl)piperazin-2-one
2-acetyl-8-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
3-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one