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N-(4-chloro-3-methoxyphenyl)-2-[3-(1H-imidazol-1-yl)pyrrolidin-1-yl]acetamide
N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carboxamide
2-(ethylamino)-N-[(8-methoxyquinolin-5-yl)methyl]-N-methylpyrimidine-5-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(4-methyl-1H-imidazol-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1'-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}spiro[indene-1,4'-piperidine]
3-(pentan-2-yl)-8-[3-(pyridin-2-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
7-cyclopentyl-2-(5-fluoropyridin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
4-[(2,4-dimethoxyphenyl)methyl]-2-(2-methylpropyl)morpholine
N-cyclohexyl-2-[(1S,5R)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
4-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
1-[(3-methylpyridin-2-yl)methyl]-4-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperazine
6-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-2-(1H-pyrazole-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(pyridin-3-yl)propan-1-one
1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-3-[3-(trifluoromethyl)benzoyl]piperidine
N-(2-chlorophenyl)-3-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]propanamide
3-{2-[6-hydroxy-4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
2-[(propan-2-yl)amino]-N-[(3,4,5-trifluorophenyl)methyl]pyrimidine-5-carboxamide
[1-(1-methylcyclopropanecarbonyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
1-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-ethoxy-2-methylpropan-1-one
(2S)-3-hydroxy-2-({5-propylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propanamide
2-methoxy-1-{1'-[2-(thiophen-3-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
2-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-6-(propan-2-yl)pyridine-3-carbonitrile
(3E)-N-(2-hydroxyethyl)-N-{[4-(methylsulfanyl)phenyl]methyl}pent-3-enamide
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}propanamide
N-(4-{[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}phenyl)cyclopropanecarboxamide
1-(butane-1-sulfonyl)-4-[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidine
3,3,3-trifluoro-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
(2S)-1-{2-chloro-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}pyrrolidine-2-carboxylic acid
(3R,4S)-1-(azepane-1-sulfonyl)-4-(propan-2-yl)pyrrolidin-3-amine
2-{2-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]-2-oxoethyl}-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2-(morpholin-4-ylmethyl)-1,4-oxazepane
6-methyl-2-({2-oxo-2-[4-(3-oxo-3,4-dihydropyrazin-2-yl)piperazin-1-yl]ethyl}sulfanyl)-3,4-dihydropyrimidin-4-one
3-(1-methyl-1H-pyrrol-2-yl)-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1H-pyrazole-5-carboxamide
N-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}methanesulfonamide
6-chloro-4-[3-(1H-imidazol-2-yl)piperidin-1-yl]quinoline
2-(dimethylamino)-7-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-amino-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1H-1,2,4-triazole-5-carboxamide
1-benzyl-8-(2-phenylethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(thiophene-2-carbonyl)piperazine
5-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-N-ethylpyrimidin-2-amine
2-(methylsulfanyl)-3-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyridine
2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)acetamide
4-(4-fluorophenoxy)-1-[2-(3-methyl-1,2-oxazol-5-yl)ethyl]piperidine
2-[1-(1H-indole-7-carbonyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
4-fluoro-N-{2-[(3-methyl-1-propyl-1H-pyrazol-4-yl)formamido]ethyl}benzamide
1-methyl-2-{2-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethyl}pyrrolidine
3-{2-oxo-2-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-1,3-oxazolidin-2-one
N-cyclooctyl-3-(1-ethyl-1H-1,2,4-triazol-5-yl)propanamide
(3S,4S)-4-cyclopropyl-1-[5-(trifluoromethyl)pyridin-2-yl]pyrrolidine-3-carboxylic acid