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5-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-3,4-dihydropyrimidin-4-one
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(furan-3-ylmethyl)pyrrolidin-3-yl]-2,6-dimethylpyrimidine-4-carboxamide
1-benzoyl-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]piperidin-4-amine
3-(azepane-1-carbonyl)-1-ethyl-N-methyl-N-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(5-fluoro-2-methylphenyl)-1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]ethan-1-one
(2S)-2-({2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazol-4-yl}formamido)propanamide
1-(3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl)-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-(1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}azetidin-3-yl)-2-methylpiperidine
6-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
1-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
3-[5-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-1,2,4-oxadiazol-3-yl]pyridine
2-(2-hydroxyethyl)-8-[3-(2-methyl-1H-1,3-benzodiazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-propoxyacetamide
2-[4-(ethoxycarbonyl)piperazin-1-yl]-2-[3-(methylsulfanyl)phenyl]acetic acid
1-[3-(2-methyl-1H-imidazol-1-yl)propyl]-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
2-benzyl-8-(4-methoxypyrimidin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
3-{2-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-[2-(3-methylthiophen-2-yl)ethyl]-2-(phenylamino)pyrimidine-5-carboxamide
N-[2-(dimethylamino)ethyl]-2-methyl-N-(oxolan-2-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
8-[2-methyl-2-(morpholin-4-yl)propyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
6-[2-(3-methoxypropyl)piperidine-1-carbonyl]quinoline
1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-2-(9-methyl-9H-carbazol-3-yl)ethan-1-one
3-(1-cyclohexylpiperidin-4-yl)-N-(3-methoxyphenyl)propanamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-(1H-pyrazol-1-yl)butanamide
[(3R,4R)-1-(5-fluoropyridin-2-yl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
1'-(cyclohex-3-ene-1-carbonyl)-5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(1S,5R)-6-(4-ethyl-5-methylthiophene-3-carbonyl)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-N-(2-methoxyethyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-(4-{[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenyl)acetamide
3-[4-(2-fluorophenyl)-1H-pyrazol-5-yl]-1-(3-phenylpropyl)piperidine
5-oxo-1-[2-oxo-6-(pyrrolidin-1-yl)-2,3-dihydro-1H-1,3-benzodiazol-5-yl]pyrrolidine-3-carboxylic acid
N-{[1-(1,3-thiazol-4-ylmethyl)piperidin-3-yl]methyl}-3-(trifluoromethyl)benzamide
6-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-N-(3-methoxypropyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
(9aR)-8-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(2-chlorophenoxy)-1-{4-[2-(pyridin-2-yl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
N,5-dimethyl-N-(2-methylpropyl)-4-{[2-(piperidin-1-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
2-[(1S,5R)-3-[(3,4-difluorophenyl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
ethyl 4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carboxylate
3-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}-1H-indazole
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-phenylpropanamide
1-(2-{1-[2-(4-methoxyphenyl)acetyl]piperidin-2-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
[2-(4-methoxyphenyl)ethyl][(2-methoxyphenyl)methyl][(1-methylpiperidin-4-yl)methyl]amine
3-{[3-(oxan-4-yl)-1-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
ethyl 3-[(4-fluorophenyl)methyl]-1-(3-methylbut-2-enoyl)piperidine-3-carboxylate
N-(pyridin-2-ylmethyl)-1-[1-(pyridine-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
4,4,4-trifluoro-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)butanamide
4-benzyl-3-[1-(oxolane-2-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
[1-(quinolin-2-yl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
ethyl 2-[(3R,4R)-3-hydroxy-4-(morpholin-4-yl)piperidin-1-yl]-1,3-oxazole-4-carboxylate