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(1s,4s)-4-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclohexan-1-ol
N-[2-(morpholin-4-yl)ethyl]-4-(4-{[2-(1H-pyrazol-1-yl)ethyl]amino}piperidin-1-yl)benzamide
N-(2,5-dimethylphenyl)-3-oxo-3-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)propanamide
[(8-methyl-2-{octahydropyrrolo[1,2-a]piperazin-2-yl}quinolin-3-yl)methyl](thiophen-2-ylmethyl)amine
N-[(3R,4R)-3-hydroxy-1-(4-methoxypyrimidin-2-yl)piperidin-4-yl]pyrazine-2-carboxamide
[3-(prop-2-en-1-yl)-1-(1,3-thiazol-2-ylmethyl)piperidin-3-yl]methanol
6-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]hexan-1-ol
1-{2-methylpyrido[2,3-d]pyrimidin-4-yl}-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
5-[2-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]pyridin-2-amine
3-[1-({1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]piperidin-4-yl}amino)ethyl]adamantan-1-ol
1-(4-tert-butylbenzoyl)-4-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)piperidine
N-(1,4-dioxan-2-ylmethyl)-7-fluoro-N-methylquinazolin-4-amine
(3S,4R)-1-(2-methoxypyridine-4-carbonyl)-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
N-{2-[1-(oxolan-3-yl)-1H-1,2,3-triazol-4-yl]quinolin-6-yl}acetamide
2-[2,4-dioxo-1-(2-phenylethyl)-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
2-({[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}amino)pyridine-3-carbonitrile
3-[(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)(methyl)amino]-1-phenylpropan-1-ol
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-[(2,3-dimethylphenyl)methyl]piperidine
1-[benzyl(methyl)amino]-3-[2-methoxy-5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)phenoxy]propan-2-ol
2-({2-[2-(furan-2-yl)phenyl]-1H-imidazol-1-yl}methyl)-3-methylpyridine
methyl[(4-methyl-1H-imidazol-5-yl)methyl]{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-N-methyl-1,3-oxazole-4-carboxamide
methyl 4-{[4-(2-chlorobenzoyl)-7-oxo-1,4-diazepan-1-yl]methyl}benzoate
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-2-(methylsulfanyl)acetamide
1-(2-chlorophenyl)-4-(5-propyl-1,3,4-oxadiazol-2-yl)piperazine
2,4-dimethoxy-5-(2-methylphenyl)pyrimidine
2-(4-chlorophenyl)-4-(4-phenyl-1H-imidazole-5-carbonyl)morpholine
2-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)-1,3-oxazole-4-carboxamide
1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-3-phenylpiperazine
1-(2-methylphenyl)-4-(pyrazine-2-carbonyl)-1,4-diazepane
4-[(diethylamino)methyl]-5-ethyl-N-(1-methoxypropan-2-yl)furan-2-carboxamide
[(3R,5R)-1-(2-fluoro-4-methylbenzoyl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
1-(2-fluorophenyl)-5-(oxolan-2-yl)-3-(2-phenylethyl)-1H-1,2,4-triazole
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}propan-1-one
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(1H-pyrazol-1-yl)butanamide
3-methyl-N-{1-[1-(3,3,3-trifluoropropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
3-[2-(2-fluorophenyl)ethyl]-1-(1,3-thiazole-4-carbonyl)piperidine
2-methoxyethyl spiro[azepane-4,2'-chromene]-1-carboxylate
3-{1-[4-hydroxy-2-(4-methylphenyl)pyrimidine-5-carbonyl]piperidin-3-yl}propanamide
methyl 4-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pentanoate
3-{3-[cyclohexyl(methyl)amino]propyl}-8-(2-hydroxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
1-{2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-({1-[2-(morpholin-4-yl)ethyl]-1H-pyrazol-4-yl}methyl)adamantan-2-amine
2-[1-(2-methylpyridin-4-yl)-1H-pyrazol-4-yl]-4-(pyrrolidine-1-carbonyl)quinoline
1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
7-methoxy-N-[(1-propyl-1H-imidazol-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(1S,3R)-N-benzyl-3-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetamido}cyclopentane-1-carboxamide
4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-5-phenyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-2-one
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-2-(2,4-dichlorophenoxy)acetamide