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3-[1-(2,6-dimethoxypyrimidin-4-yl)piperidin-3-yl]-N-(4-methoxy-2-methylphenyl)propanamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N,2,4-trimethylpyrimidine-5-carboxamide
methyl 5-[(3E)-4-phenylbut-3-enoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-4-(1H-imidazol-2-yl)piperidine
2-({methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)benzoic acid
4-(4-methoxyphenoxymethyl)-1-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperidine
9-(6-methylpyrimidin-4-yl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-({[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
methyl (2S)-1-{2-[4-(4-{[2-(1H-pyrazol-1-yl)ethyl]amino}piperidin-1-yl)phenyl]acetyl}pyrrolidine-2-carboxylate
N-({1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]piperidin-3-yl}methyl)acetamide
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-(5-methoxy-1,2-dimethyl-1H-indole-3-carbonyl)pyrrolidin-3-yl]methanol
5-(2-chlorophenyl)-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]furan-2-carboxamide
methyl 2-(5-aminopyrazin-2-yl)benzoate
3-{[(2,3-difluoro-4-methoxyphenyl)methyl]amino}-N-(furan-2-ylmethyl)propanamide
5-(1H-1,3-benzodiazol-1-yl)-6-methylpyridin-2-amine
2-(2-ethyl-1H-imidazol-1-yl)-1-{2-[(3-fluorophenyl)methyl]morpholin-4-yl}ethan-1-one
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-{2-oxo-2-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3S,5R,9R)-11-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-5-hydroxy-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
N,5-dimethyl-4-(1-methyl-1H-pyrazol-4-yl)-N-[(3-methylthiophen-2-yl)methyl]pyrimidin-2-amine
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-2-phenylacetamide
6-{3-[(4-phenyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-9H-purine
(1-{[5-(4-methylpiperazine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}piperidin-4-yl)methanol
4-(2,3-dimethylquinoxaline-6-amido)oxane-4-carboxylic acid
3-(4-methoxy-2-methylbenzoyl)-1-(thiophene-2-sulfonyl)piperidine
N-[3-(1H-imidazol-1-yl)propyl]-3-(pyridin-4-yl)propanamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(dimethyl-1,3-thiazole-5-carbonyl)piperidine
[(2S,4R)-1-{[2-(butylsulfanyl)pyrimidin-5-yl]methyl}-4-(dimethylamino)pyrrolidin-2-yl]methanol
6-methyl-4-oxo-1-(oxolan-2-ylmethyl)-2-(2-phenylethyl)-N-(quinolin-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
5-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-2-(4-methylphenyl)pyrimidin-4-ol
N,N-diethyl-2-[1-(2-hydroxyethyl)-1H-pyrazol-4-yl]-7,8-dimethylquinoline-4-carboxamide
5-(2-methoxypyridin-3-yl)thiophene-2-sulfonamide
2-[4-(ethoxycarbonyl)piperazin-1-yl]-2-(furan-3-yl)acetic acid
N-[(3-methoxyphenyl)methyl]-2-oxo-N-(prop-2-en-1-yl)-2-(pyrrolidin-1-yl)acetamide
3-{[2-(2-phenyl-1,3-oxazol-4-yl)-1H-imidazol-1-yl]methyl}-5-(propan-2-yl)-1,2,4-oxadiazole
N-[3-(pyridin-2-yl)propyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
(4aS,8aR)-1-(2-aminoethyl)-6-(1H-1,2,3-benzotriazole-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-(2-methoxyethyl)-2-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-1,2,3,4-tetrahydroisoquinoline-8-sulfonamide
N-(butan-2-yl)-N-ethyl-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
[4-({2-[(oxolan-2-ylmethyl)amino]pyrimidin-5-yl}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methanol
(5S,9aS,9bS)-2-[(2-methoxyphenyl)methyl]-5-[5-(propan-2-yl)-1H-pyrazol-3-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-methyl-8-(quinoline-3-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{1-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-(pyridin-3-yloxy)acetamide
1-{4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
1-[3-(1H-imidazol-2-yl)propyl]-5-methyl-5-phenylpiperidin-2-one
8-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}quinoline
2-(1-{[3-(difluoromethoxy)phenyl]methyl}-1H-1,2,3-triazol-4-yl)-5-ethylpyridine
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}acetic acid
N-[2-methyl-6-(propan-2-yl)phenyl]-2-{[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]amino}acetamide
1-(pyridin-4-ylmethyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol