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1-propyl-5-[3-(1H-pyrazol-1-yl)azetidin-1-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
9-(6-cyclopropylpyrimidin-4-yl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(4,6-dimethylpyrimidin-2-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-[2-(dimethylamino)ethyl]-3-(2-fluorophenyl)-3-{2-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)cyclopent-3-ene-1-carboxamide
4-[3-(azocan-1-yl)propanoyl]-1-(4-chlorophenyl)-5-methylpiperazin-2-one
(4aS,8aR)-6-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
(1R,3S,5S)-8-[5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carbonyl]-8-azabicyclo[3.2.1]octan-3-ol
1-(4-{[(cyclohexylmethyl)amino]methyl}-2-methoxyphenoxy)-3-(4-ethylpiperazin-1-yl)propan-2-ol
4-{[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]methyl}-1-ethyl-1H-pyrrole-2-carbonitrile
3-{5-[2-(2,3-dimethylphenoxy)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
5-(6-methoxypyrimidin-4-yl)-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-phenyl-1H-1,2,3-triazole-5-carboxamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)thiophene-3-carboxamide
3-(2-methoxyethyl)-1-[3-(pyridin-3-yl)propanoyl]piperidine-3-carboxylic acid
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]pyridin-2-amine
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-{[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
3,5-dimethyl-2-{3-[(methylsulfanyl)methyl]piperidine-1-carbonyl}-1H-indole
N-{[3-(4-fluorophenyl)oxolan-3-yl]methyl}-2-(2,3,6-trimethylphenoxy)acetamide
1-methyl-9-[3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanoyl]-1,4,9-triazaspiro[5.5]undecan-5-one
4-phenoxy-1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidine-4-carboxylic acid
8-(5-amino-1H-pyrazole-3-carbonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{1-[1-(3-chloro-4-fluorobenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
2-{methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}-2-{4-[(pyrrolidine-1-carbonyl)amino]phenyl}acetic acid
1,3-dimethyl-N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-1H-pyrazole-5-carboxamide
7-[2-(3-chlorophenyl)-1H-imidazol-1-yl]-4-methyl-3,4-dihydro-2H-1,4-benzoxazin-3-one
1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(thiophen-3-yl)propan-1-one
4-{[3-(3-phenylpropanoyl)piperidin-1-yl]methyl}benzamide
4-[1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperidine-4-carbonyl]morpholine
N-(pyridin-4-ylmethyl)-4-[5-(trifluoromethyl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
4-[(2-methylpyridin-3-yl)oxy]-1-(thiophene-2-carbonyl)piperidine-4-carboxylic acid
7-amino-4-[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one
3-propyl-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(2,6-dichlorobenzoyl)piperidine
2-(2,3-dihydro-1H-isoindol-2-yl)-N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]acetamide
N-[(3-chloro-2-fluorophenyl)methyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
(3S,4R)-1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
5-chloro-3-ethyl-4-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}-1-methyl-1H-pyrazole
N-cyclooctyl-2-({[1-(hydroxymethyl)cyclobutyl]methyl}amino)acetamide
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-3-(1H-pyrazol-5-yl)piperidine
2-{4-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-ylmethyl]phenyl}-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
N-ethyl-N-(oxan-4-yl)-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
N-[3-({ethyl[(1-methylpyrrolidin-3-yl)methyl]carbamoyl}amino)phenyl]butanamide
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]pyrrolidine-1-sulfonamide
2-{5-[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetic acid
N-[(2R,3R)-1'-[2-(cyclohex-1-en-1-yl)acetyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-{2-[3-(trifluoromethyl)phenyl]ethyl}propanamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-ethylpyrimidin-2-amine
6-ethyl-N-[2-(2-fluorophenyl)ethyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine